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Target
Mu-type opioid receptor
Ligand
BDBM50083734
Substrate
n/a
Meas. Tech.
ChEMBL_136095 (CHEMBL745617)
IC50
0.110000±n/a nM
Citation
 Burden, JE; Davis, P; Porreca, F; Spatola, AF Synthesis and biological activities of position one and three transposed analogs of the opioid peptide YKFA. Bioorg Med Chem Lett 9:3441-6 (2000) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50083734
Synonyms:
2-Amino-N-[(R)-6-(4-hydroxy-benzyl)-3-methyl-2,5,8-trioxo-1,4,7triaza-cyclotridec-9-yl]-3-phenyl-propionamide | CHEMBL2370485
Type:
Small organic molecule
Emp. Form.:
C27H35N5O5
Mol. Mass.:
509.5973
SMILES:
C[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CCCCNC1=O)NC(=O)[C@@H](N)Cc1ccc(O)cc1
Structure:
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