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Target
Bacterial leucyl aminopeptidase
Ligand
BDBM50129202
Substrate
n/a
Meas. Tech.
ChEBML_98920
Ki
350±n/a nM
Citation
 Stoermer, D; Liu, Q; Hall, MR; Flanary, JM; Thomas, AG; Rojas, C; Slusher, BS; Tsukamoto, T Synthesis and biological evaluation of hydroxamate-Based inhibitors of glutamate carboxypeptidase II. Bioorg Med Chem Lett 13:2097-100 (2003) [PubMed]  Article 
Target
Name:
Bacterial leucyl aminopeptidase
Synonyms:
AMPX_VIBPR | Bacterial leucyl aminopeptidase precursor
Type:
PROTEIN
Mol. Mass.:
54213.72
Organism:
Vibrio proteolyticus
Description:
ChEMBL_1507540
Residue:
504
Sequence:
MKYTKTLLAMVLSATFCQAYAEDKVWISIGADANQTVMKSGAESILPNSVASSGQVWVGQVDVAQLAELSHNMHEEHNRCGGYMVHPSAQSAMAASAMPTTLASFVMPPITQQATVTAWLPQVDASQITGTISSLESFTNRFYTTTSGAQASDWIASEWQALSASLPNASVKQVSHSGYNQKSVVMTITGSEAPDEWIVIGGHLDSTIGSHTNEQSVAPGADDDASGIAAVTEVIRVLSENNFQPKRSIAFMAYAAEEVGLRGSQDLANQYKSEGKNVVSALQLDMTNYKGSAQDVVFITDYTDSNFTQYLTQLMDEYLPSLTYGFDTCGYACSDHASWHNAGYPAAMPFESKFNDYNPRIHTTQDTLANSDPTGSHAKKFTQLGLAYAIEMGSATGDTPTPGNQLEDGVPVTDLSGSRGSNVWYTFELETQKNLQITTSGGYGDLDLYVKFGSKASKQNWDCRPYLSGNNEVCTFNNASPGTYSVMLTGYSNYSGASLKASTF
  
Inhibitor
Name:
BDBM50129202
Synonyms:
(S)-2-Amino-4-methyl-pentanoic acid hydroxyamide | (S)-2-amino-N-hydroxy-4-methylpentanamide | CHEMBL303296 | L-LEUCYL-HYDROXYLAMINE
Type:
Small organic molecule
Emp. Form.:
C6H14N2O2
Mol. Mass.:
146.1876
SMILES:
CC(C)C[C@H](N)C(=O)NO
Structure:
Search PDB for entries with ligand similarity: