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Target
Elongin-C
Ligand
BDBM50590276
Substrate
n/a
Meas. Tech.
ChEMBL_2195889 (CHEMBL5108405)
Ki
397±n/a nM
Citation
de Castro, GV; Ciulli, A Estimating the cooperativity of PROTAC-induced ternary complexes using RSC Med Chem 12:1765-1770 (2021) [PubMed]
More Info.:
Target
Name:
Elongin-C
Synonyms:
ELOC | ELOC_HUMAN | Elongin 15 kDa subunit | Elongin-C | RNA polymerase II transcription factor SIII subunit C | SIII p15 | TCEB1 | Transcription elongation factor B polypeptide 1
Type:
PROTEIN
Mol. Mass.:
12466.49
Organism:
Homo sapiens (Human)
Description:
ChEMBL_108414
Residue:
112
Sequence:
MDGEEKTYGGCEGPDAMYVKLISSDGHEFIVKREHALTSGTIKAMLSGPGQFAENETNEVNFREIPSHVLSKVCMYFTYKVRYTNSSTEIPEFPIAPEIALELLMAANFLDC