Target
Bacterial leucyl aminopeptidase
Ligand
BDBM50336495
Substrate
n/a
Meas. Tech.
ChEMBL_766295 (CHEMBL1826227)
Ki
900000±n/a nM
Citation
 Maiereanu, CSchmitt, CSchifano-Faux, NLe Nouën, DDefoin, ATarnus, C A novel amino-benzosuberone derivative is a picomolar inhibitor of mammalian aminopeptidase N/CD13. Bioorg Med Chem 19:5716-33 (2011) [PubMed]  Article 
Target
Name:
Bacterial leucyl aminopeptidase
Synonyms:
AMPX_VIBPR | Bacterial leucyl aminopeptidase precursor
Type:
PROTEIN
Mol. Mass.:
54213.72
Organism:
Vibrio proteolyticus
Description:
ChEMBL_1507540
Residue:
504
Sequence:
MKYTKTLLAMVLSATFCQAYAEDKVWISIGADANQTVMKSGAESILPNSVASSGQVWVGQVDVAQLAELSHNMHEEHNRCGGYMVHPSAQSAMAASAMPTTLASFVMPPITQQATVTAWLPQVDASQITGTISSLESFTNRFYTTTSGAQASDWIASEWQALSASLPNASVKQVSHSGYNQKSVVMTITGSEAPDEWIVIGGHLDSTIGSHTNEQSVAPGADDDASGIAAVTEVIRVLSENNFQPKRSIAFMAYAAEEVGLRGSQDLANQYKSEGKNVVSALQLDMTNYKGSAQDVVFITDYTDSNFTQYLTQLMDEYLPSLTYGFDTCGYACSDHASWHNAGYPAAMPFESKFNDYNPRIHTTQDTLANSDPTGSHAKKFTQLGLAYAIEMGSATGDTPTPGNQLEDGVPVTDLSGSRGSNVWYTFELETQKNLQITTSGGYGDLDLYVKFGSKASKQNWDCRPYLSGNNEVCTFNNASPGTYSVMLTGYSNYSGASLKASTF
  
Inhibitor
Name:
BDBM50336495
Synonyms:
7-Amino-5,7,8,9-tetrahydro-benzocyclohepten-6-one, hydrochloride | CHEMBL1668626
Type:
Small organic molecule
Emp. Form.:
C11H13NO
Mol. Mass.:
175.227
SMILES:
NC1CCc2ccccc2CC1=O
Structure:
Search PDB for entries with ligand similarity: