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Target
Tissue alpha-L-fucosidase
Ligand
BDBM50242419
Substrate
n/a
Meas. Tech.
ChEMBL_216279 (CHEMBL819885)
Ki
300000±n/a nM
Citation
 Witczak, ZJ; Sun, J; Mielguj, R Synthesis of L-fucopyranosyl-4-thiodisaccharides from levoglucosenone and their inhibitory activity on -L-fucosidase Bioorg Med Chem Lett 5:2169-2174 (1995)    Article 
Target
Name:
Tissue alpha-L-fucosidase
Synonyms:
Alpha-L-fucosidase I | Alpha-L-fucoside fucohydrolase | FUCA1 | FUCO_HUMAN | Tissue alpha-L-fucosidase
Type:
PROTEIN
Mol. Mass.:
53690.69
Organism:
Homo sapiens (Human)
Description:
ChEMBL_34088
Residue:
466
Sequence:
MRAPGMRSRPAGPALLLLLLFLGAAESVRRAQPPRRYTPDWPSLDSRPLPAWFDEAKFGVFIHWGVFSVPAWGSEWFWWHWQGEGRPQYQRFMRDNYPPGFSYADFGPQFTARFFHPEEWADLFQAAGAKYVVLTTKHHEGFTNWPSPVSWNWNSKDVGPHRDLVGELGTALRKRNIRYGLYHSLLEWFHPLYLLDKKNGFKTQHFVSAKTMPELYDLVNSYKPDLIWSDGEWECPDTYWNSTNFLSWLYNDSPVKDEVVVNDRWGQNCSCHHGGYYNCEDKFKPQSLPDHKWEMCTSIDKFSWGYRRDMALSDVTEESEIISELVQTVSLGGNYLLNIGPTKDGLIVPIFQERLLAVGKWLSINGEAIYASKPWRVQWEKNTTSVWYTSKGSAVYAIFLHWPENGVLNLESPITTSTTKITMLGIQGDLKWSTDPDKGLFISLPQLPPSAVPAEFAWTIKLTGVK
  
Inhibitor
Name:
BDBM50242419
Synonyms:
6-Deoxy-L-galactose | 6-deoxy-L-galactopyranoseL-fucopyranose | CHEMBL469449 | L-fucopyranose | L-fucose
Type:
Small organic molecule
Emp. Form.:
C6H12O5
Mol. Mass.:
164.1565
SMILES:
C[C@@H]1OC(O)[C@@H](O)[C@H](O)[C@@H]1O |r|
Structure:
Search PDB for entries with ligand similarity: