Reaction Details Report a problem with these data
Target
Cannabinoid receptor 2
Ligand
BDBM50263073
Substrate
n/a
Meas. Tech.
ChEMBL_490517 (CHEMBL981123)
Ki
>7900±n/a nM
Citation
 Urbani, P; Cascio, MG; Ramunno, A; Bisogno, T; Saturnino, C; Di Marzo, V Novel sterically hindered cannabinoid CB1 receptor ligands. Bioorg Med Chem 16:7510-5 (2008) [PubMed]  Article 
Target
Name:
Cannabinoid receptor 2
Synonyms:
CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
39690.94
Organism:
Homo sapiens (Human)
Description:
P34972
Residue:
360
Sequence:
MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILSSHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTASVGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCSELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLDVRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYALRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
  
Inhibitor
Name:
BDBM50263073
Synonyms:
2-(4-Chlorophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide | CHEMBL475909
Type:
Small organic molecule
Emp. Form.:
C29H26ClNO
Mol. Mass.:
439.976
SMILES:
Clc1ccc(cc1)C(C(=O)NCCC(c1ccccc1)c1ccccc1)c1ccccc1
Structure:
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