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Target
Solute carrier family 15 member 2
Ligand
BDBM17658
Substrate
n/a
Meas. Tech.
ChEMBL_836021 (CHEMBL2077253)
IC50
3000000±n/a nM
Citation
 Wang, H; Fei, YJ; Ganapathy, V; Leibach, FH Electrophysiological characteristics of the proton-coupled peptide transporter PEPT2 cloned from rat brain. Am J Physiol 275:967-75 (1998) [PubMed]  Article 
Target
Name:
Solute carrier family 15 member 2
Synonyms:
Oligopeptide transporter, kidney isoform | Pept2 | S15A2_RAT | Slc15a2
Type:
PROTEIN
Mol. Mass.:
81331.63
Organism:
Rattus norvegicus
Description:
ChEMBL_838253
Residue:
729
Sequence:
MNPFQKNESKETLFSPVSTEEMLPRPPSPPKKSPPKIFGSSYPVSIAFIVVNEFCERFSYYGMKAVLTLYFLYFLHWNEDTSTSVYHAFSSLCYFTPILGAAIADSWLGKFKTIIYLSLVYVLGHVFKSLGAIPILGGKMLHTILSLVGLSLIALGTGGIKPCVAAFGGDQFEEEHAEARTRYFSVFYLAINAGSLISTFITPMLRGDVKCFGQDCYALAFGVPGLLMVLALVVFAMGSKMYRKPPPEGNIVAQVIKCIWFALCNRFRNRSGDLPKRQHWLDWAAEKYPKHLIADVKALTRVLFLYIPLPMFWALLDQQGSRWTLQANKMNGDLGFFVLQPDQMQVLNPFLVLIFIPLFDLVIYRLISKCRINFSSLRKMAVGMILACLAFAVAALVETKINGMIHPQPASQEIFLQVLNLADGDVKVTVLGSRNNSLLVESVSSFQNTTHYSKLHLEAKSQDLHFHLKYNSLSVHNDHSVEEKNCYQLLIHQDGESISSMLVKDTGIKPANGMAAIRFINTLHKDLNISLDTDAPLSVGKDYGVSAYRTVLRGKYPAVHCETEDKVFSLDLGQLDFGTTYLFVITNITSQGLQAWKAEDIPVNKLSIAWQLPQYVLVTAAEVMFSVTGLEFSYSQAPSSMKSVLQAAWLLTVAVGNIIVLVVAQFSGLAQWAEFVLFSCLLLVVCLIFSVMAYYYVPLKSEDTREATDKQIPAVQGNMINLETKNTRL
  
Inhibitor
Name:
BDBM17658
Synonyms:
(2S)-2-[(3S)-3-acetamido-3-formamidopropanoic acid]pentanedioic acid | N-acetylaspartylglutamate (NAAG) | NAAG | [3H]NAAG
Type:
Small organic molecule
Emp. Form.:
C11H16N2O8
Mol. Mass.:
304.2533
SMILES:
CC(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CCC(O)=O)C(O)=O |r|
Structure:
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