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Target
Histamine H2 receptor
Ligand
BDBM22881
Substrate
n/a
Meas. Tech.
ChEBML_85683
Kd
11482±n/a nM
Citation
 van der Goot, H; Eriks, JC; Leurs, R; Timmerman, H Amselamine, a new selective histamine H2-receptor agonist Bioorg Med Chem Lett 4:1913-1916 (1994)    Article 
Target
Name:
Histamine H2 receptor
Synonyms:
Gastric receptor I | H2R | HISTAMINE H2 | HRH2_RAT | Hrh2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40269.37
Organism:
RAT
Description:
HISTAMINE H2 HRH2 RAT::P25102
Residue:
358
Sequence:
MEPNGTVHSCCLDSMALKVTISVVLTTLILITIAGNVVVCLAVSLNRRLRSLTNCFIVSLAATDLLLGLLVLPFSAIYQLSFTWSFGHVFCNIYTSLDVMLCTASILNLFMISLDRYCAVTDPLRYPVLVTPVRVAISLVFIWVISITLSFLSIHLGWNSRNGTRGGNDTFKCKVQVNEVYGLVDGLVTFYLPLLIMCVTYYRIFKIAREQAKRINHISSWKAATIREHKATVTLAAVMGAFIICWFPYFTAFVYRGLRGDDAINEAVEGIVLWLGYANSALNPILYAALNRDFRTAYQQLFHCKFASHNSHKTSLRLNNSLLPRSQSREGRWQEEKPLKLQVWSGTELTHPQGNPIR
  
Inhibitor
Name:
BDBM22881
Synonyms:
5-(2-aminoethyl)-4-methyl-1,3-thiazol-2-amine | Amthamine | CHEMBL554964
Type:
Small organic molecule
Emp. Form.:
C6H11N3S
Mol. Mass.:
157.237
SMILES:
Cc1nc(N)sc1CCN
Structure:
Search PDB for entries with ligand similarity: