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Target
Urotensin-2
Ligand
BDBM50416339
Substrate
n/a
Meas. Tech.
ChEMBL_643307 (CHEMBL1177478)
EC50
724.44±n/a nM
Citation
 Lehmann, F; Currier, EA; Olsson, R; Ma, JN; Burstein, ES; Hacksell, U; Luthman, K Optimization of isochromanone based urotensin II receptor agonists. Bioorg Med Chem 18:4844-54 (2011) [PubMed]  Article 
Target
Name:
Urotensin-2
Synonyms:
UTS2 | UTS2_HUMAN
Type:
PROTEIN
Mol. Mass.:
14297.49
Organism:
Homo sapiens (Human)
Description:
ChEMBL_643307
Residue:
124
Sequence:
MYKLASCCLLFIGFLNPLLSLPLLDSREISFQLSAPHEDARLTPEELERASLLQILPEMLGAERGDILRKADSSTNIFNPRGNLRKFQDFSGQDPNILLSHLLARIWKPYKKRETPDCFWKYCV
  
Inhibitor
Name:
BDBM50416339
Synonyms:
CHEMBL1173081
Type:
Small organic molecule
Emp. Form.:
C25H29ClN2O2
Mol. Mass.:
424.963
SMILES:
CN(C)CCC1(Cc2cc(ccc2C(=O)O1)N(CC=C)CC=C)c1ccc(Cl)cc1
Structure:
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