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Target
Solute carrier family 22 member 16
Ligand
BDBM50037268
Substrate
n/a
Meas. Tech.
ChEMBL_838411 (CHEMBL2076433)
Ki
30000±n/a nM
Citation
 Enomoto, A; Wempe, MF; Tsuchida, H; Shin, HJ; Cha, SH; Anzai, N; Goto, A; Sakamoto, A; Niwa, T; Kanai, Y; Anders, MW; Endou, H Molecular identification of a novel carnitine transporter specific to human testis. Insights into the mechanism of carnitine recognition. J Biol Chem 277:36262-71 (2002) [PubMed]  Article 
Target
Name:
Solute carrier family 22 member 16
Synonyms:
CT2 | Carnitine transporter 2 | FLIPT2 | Flipt 2 | Fly-like putative transporter 2 | OCT6 | Organic cation transporter OKB1 | Organic cation/carnitine transporter 6 | S22AG_HUMAN | SLC22A16
Type:
PROTEIN
Mol. Mass.:
64624.46
Organism:
Homo sapiens (Human)
Description:
ChEMBL_838411
Residue:
577
Sequence:
MGSRHFEGIYDHVGHFGRFQRVLYFICAFQNISCGIHYLASVFMGVTPHHVCRPPGNVSQVVFHNHSNWSLEDTGALLSSGQKDYVTVQLQNGEIWELSRCSRNKRENTSSLGYEYTGSKKEFPCVDGYIYDQNTWKSTAVTQWNLVCDRKWLAMLIQPLFMFGVLLGSVTFGYFSDRLGRRVVLWATSSSMFLFGIAAAFAVDYYTFMAARFFLAMVASGYLVVGFVYVMEFIGMKSRTWASVHLHSFFAVGTLLVALTGYLVRTWWLYQMILSTVTVPFILCCWVLPETPFWLLSEGRYEEAQKIVDIMAKWNRASSCKLSELLSLDLQGPVSNSPTEVQKHNLSYLFYNWSITKRTLTVWLIWFTGSLGFYSFSLNSVNLGGNEYLNLFLLGVVEIPAYTFVCIAMDKVGRRTVLAYSLFCSALACGVVMVIPQKHYILGVVTAMVGKFAIGAAFGLIYLYTAELYPTIVRSLAVGSGSMVCRLASILAPFSVDLSSIWIFIPQLFVGTMALLSGVLTLKLPETLGKRLATTWEEAAKLESENESKSSKLLLTTNNSGLEKTEAITPRDSGLGE
  
Inhibitor
Name:
BDBM50037268
Synonyms:
(-)-Carnitine | (-)-L-Carnitine | (3R)-3-hydroxy-4-(trimethylammonio)butanoate | (R)-Carnitine | CHEMBL1149 | Carnitine | LEVOCARNITINE
Type:
Small organic molecule
Emp. Form.:
C7H15NO3
Mol. Mass.:
161.1989
SMILES:
C[N+](C)(C)C[C@H](O)CC([O-])=O |r|
Structure:
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