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Target
Solute carrier organic anion transporter family member 2A1
Ligand
BDBM50390979
Substrate
n/a
Meas. Tech.
ChEMBL_836139 (CHEMBL2077575)
Ki
5800±n/a nM
Citation
 Kanai, N; Lu, R; Satriano, JA; Bao, Y; Wolkoff, AW; Schuster, VL Identification and characterization of a prostaglandin transporter. Science 268:866-869 (1995) [PubMed]  Article 
Target
Name:
Solute carrier organic anion transporter family member 2A1
Synonyms:
Matr1 | Matrin F/G 1 | Prostaglandin transporter (PGT) | SO2A1_RAT | Slc21a2 | Slco2a1 | Solute carrier family 21 member 2
Type:
Protein
Mol. Mass.:
70404.97
Organism:
Rattus norvegicus (Rat)
Description:
Q00910
Residue:
644
Sequence:
MGLLLKPGARQGSGTSSVPDRRCPRSVFSNIKVFVLCHGLLQLCQLLYSAYFKSSLTTIEKRFGLSSSSSGLISSLNEISNATLIIFISYFGSRVNRPRMIGIGGLLLAAGAFVLTLPHFLSEPYQYTSTTDGNRSSFQTDLCQKHFGALPPSKCHSTVPDTHKETSSLWGLMVVAQLLAGIGTVPIQPFGISYVDDFAEPTNSPLYISILFAIAVFGPAFGYLLGSVMLRIFVDYGRVDTATVNLSPGDPRWIGAWWLGLLISSGFLIVTSLPFFFFPRAMSRGAERSVTAEETMQTEEDKSRGSLMDFIKRFPRIFLRLLMNPLFMLVVLSQCTFSSVIAGLSTFLNKFLEKQYGATAAYANFLIGAVNLPAAALGMLFGGILMKRFVFPLQTIPRVAATIITISMILCVPLFFMGCSTSAVAEVYPPSTSSSIHPQQPPACRRDCSCPDSFFHPVCGDNGVEYVSPCHAGCSSTNTSSEASKEPIYLNCSCVSGGSASAKTGSCPTSCAQLLLPSIFLISFAALIACISHNPLYMMVLRVVNQDEKSFAIGVQFLLMRLLAWLPAPSLYGLLIDSSCVRWNYLCSGRRGACAYYDNDALRNRYLGLQMVYKALGTLLLFFISWRMKKNREYSLQENTSGLI
  
Inhibitor
Name:
BDBM50390979
Synonyms:
BROMOSULFOPHTHALEIN
Type:
Small organic molecule
Emp. Form.:
C20H8Br4O10S2
Mol. Mass.:
792.019
SMILES:
Oc1ccc(cc1S([O-])(=O)=O)C1(OC(=O)c2c1c(Br)c(Br)c(Br)c2Br)c1ccc(O)c(c1)S([O-])(=O)=O
Structure:
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