Reaction Details Report a problem with these data
Target
Phosphoglycerate mutase 1
Ligand
BDBM50103572
Substrate
n/a
Meas. Tech.
ChEMBL_1435601 (CHEMBL3386524)
Ki
3910±n/a nM
Citation
Granchi, C; Fancelli, D; Minutolo, F An update on therapeutic opportunities offered by cancer glycolytic metabolism. Bioorg Med Chem Lett 24:4915-25 (2014) [PubMed] Article
More Info.:
Target
Name:
Phosphoglycerate mutase 1
Synonyms:
BPG-dependent PGAM 1 | PGAM-B | PGAM1 | PGAM1_HUMAN | PGAMA | Phosphoglycerate mutase 1 | Phosphoglycerate mutase isozyme B
Type:
PROTEIN
Mol. Mass.:
28806.11
Organism:
Homo sapiens (Human)
Description:
ChEMBL_109479
Residue:
254
Sequence:
MAAYKLVLIRHGESAWNLENRFSGWYDADLSPAGHEEAKRGGQALRDAGYEFDICFTSVQKRAIRTLWTVLDAIDQMWLPVVRTWRLNERHYGGLTGLNKAETAAKHGEAQVKIWRRSYDVPPPPMEPDHPFYSNISKDRRYADLTEDQLPSCESLKDTIARALPFWNEEIVPQIKEGKRVLIAAHGNSLRGIVKHLEGLSEEAIMELNLPTGIPIVYELDKNLKPIKPMQFLGDEETVRKAMEAVAAQGKAKK