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Target
Vasoactive intestinal polypeptide receptor 1
Ligand
BDBM50435130
Substrate
n/a
Meas. Tech.
ChEMBL_1559802 (CHEMBL3776015)
IC50
0.110±n/a nM
Citation
 Waszkielewicz, AM; Gunia-Krzyzak, A; Powroznik, B; Sloczynska, K; Pekala, E; Walczak, M; Bednarski, M; Zeslawska, E; Nitek, W; Marona, H Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents. Bioorg Med Chem 24:1793-810 (2016) [PubMed]  Article 
Target
Name:
Vasoactive intestinal polypeptide receptor 1
Synonyms:
VIP 1 | VIPR1 | VIPR1_HUMAN | Vasoactive intestinal polypeptide receptor 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
51557.18
Organism:
Homo sapiens (Human)
Description:
VIP 1 VIPR1 0::P32241
Residue:
457
Sequence:
MRPPSPLPARWLCVLAGALAWALGPAGGQAARLQEECDYVQMIEVQHKQCLEEAQLENETIGCSKMWDNLTCWPATPRGQVVVLACPLIFKLFSSIQGRNVSRSCTDEGWTHLEPGPYPIACGLDDKAASLDEQQTMFYGSVKTGYTIGYGLSLATLLVATAILSLFRKLHCTRNYIHMHLFISFILRAAAVFIKDLALFDSGESDQCSEGSVGCKAAMVFFQYCVMANFFWLLVEGLYLYTLLAVSFFSERKYFWGYILIGWGVPSTFTMVWTIARIHFEDYGCWDTINSSLWWIIKGPILTSILVNFILFICIIRILLQKLRPPDIRKSDSSPYSRLARSTLLLIPLFGVHYIMFAFFPDNFKPEVKMVFELVVGSFQGFVVAILYCFLNGEVQAELRRKWRRWHLQGVLGWNPKYRHPSGGSNGATCSTQVSMLTRVSPGARRSSSFQAEVSLV
  
Inhibitor
Name:
BDBM50435130
Synonyms:
CHEMBL1893324
Type:
Small organic molecule
Emp. Form.:
C147H238N44O42S
Mol. Mass.:
3325.797
SMILES:
n/a
Structure:
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