Reaction Details Report a problem with these data
Target
Neurotensin
Ligand
BDBM82479
Substrate
n/a
Ki
1000±n/a nM
Comments
PDSP_1408
Citation
 Schotte, A; Janssen, PF; Gommeren, W; Luyten, WH; Van Gompel, P; Lesage, AS; De Loore, K; Leysen, JE Risperidone compared with new and reference antipsychotic drugs: in vitro and in vivo receptor binding. Psychopharmacology (Berl) 124:57-73 (1996) [PubMed]  Article 
Target
Name:
Neurotensin
Synonyms:
NEUT_CAVPO | NT | NTS | Neurotensin
Type:
Enzyme Catalytic Domain
Mol. Mass.:
1681.93
Organism:
GUINEA PIG
Description:
NT 0 GUINEA PIG::P32560
Residue:
13
Sequence:
QLYENKSRRPYIL
  
Inhibitor
Name:
BDBM82479
Synonyms:
CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE49340, Rank 2
Type:
Small organic molecule
Emp. Form.:
C17H20N4S
Mol. Mass.:
312.432
SMILES:
CN1CCN(CC1)C1=c2cc(C)sc2=Nc2ccccc2N1 |c:8,15|
Structure:
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