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Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96584
Substrate
n/a
EC50
>29913±n/a nM
Citation
 PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 agonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G protein alpha 16 | G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | Guanine nucleotide-binding protein subunit alpha-15 [Y147C]
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRACYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96584
Synonyms:
4-[(2,3-dihydro-1,4-benzodioxin-3-ylmethylamino)methylene]cyclohexa-2,5-dien-1-one | 4-[(2,3-dihydro-1,4-benzodioxin-3-ylmethylamino)methylidene]-1-cyclohexa-2,5-dienone | 4-[(2,3-dihydro-1,4-benzodioxin-3-ylmethylamino)methylidene]cyclohexa-2,5-dien-1-one | MLS000106702 | SMR000111079 | cid_5340822
Type:
Small organic molecule
Emp. Form.:
C16H15NO3
Mol. Mass.:
269.2952
SMILES:
Oc1ccc(C=NCC2COc3ccccc3O2)cc1 |w:6.6|
Structure:
Search PDB for entries with ligand similarity: