Reaction Details Report a problem with these data
Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96825
Substrate
n/a
EC50
>29940±n/a nM
Citation
 PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 agonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G protein alpha 16 | G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | Guanine nucleotide-binding protein subunit alpha-15 [Y147C]
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRACYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96825
Synonyms:
(2-methoxy-6-methyl-phenyl)-(2-oxazolin-2-yl)amine | MLS003106542 | N-(2-methoxy-6-methyl-phenyl)-4,5-dihydro-1,3-oxazol-2-amine | N-(2-methoxy-6-methylphenyl)-4,5-dihydro-1,3-oxazol-2-amine | N-(2-methoxy-6-methylphenyl)-4,5-dihydrooxazol-2-amine | SMR001821441 | cid_98724
Type:
Small organic molecule
Emp. Form.:
C11H14N2O2
Mol. Mass.:
206.2411
SMILES:
COc1cccc(C)c1N=C1NCCO1 |w:9.9|
Structure:
Search PDB for entries with ligand similarity: