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Target
Galectin-3
Ligand
BDBM120770
Substrate
n/a
Meas. Tech.
Fluorescence Polarization-Based Assay
Kd
430±n/a nM
Citation
 Leffler, H; Nilsson, UJ; Von Wachenfeldt, H Galactoside inhibitors of galectins US Patent  US8703720 Publication Date 4/22/2014 
Target
Name:
Galectin-3
Synonyms:
LEG3_HUMAN | LGALS3 | MAC2
Type:
Enzyme
Mol. Mass.:
26156.54
Organism:
Homo sapiens (Human)
Description:
P17931
Residue:
250
Sequence:
MADNFSLHDALSGSGNPNPQGWPGAWGNQPAGAGGYPGASYPGAYPGQAPPGAYPGQAPPGAYPGAPGAYPGAPAPGVYPGPPSGPGAYPSSGQPSATGAYPATGPYGAPAGPLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI
  
Inhibitor
Name:
BDBM120770
Synonyms:
US8703720, 7
Type:
Small organic molecule
Emp. Form.:
C24H38N8O8
Mol. Mass.:
566.6073
SMILES:
CCCNC(=O)c1cn(nn1)C1CCC[C@@H](O[C@@H]2OC(CO)[C@H](O)[C@@H](C2O)n2cc(nn2)C(=O)NCCC)C1O |r|
Structure:
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