Reaction Details Report a problem with these data
Target
Sphingosine 1-phosphate receptor 2
Ligand
BDBM149712
Substrate
n/a
Meas. Tech.
Fluorescence-Based Assay
pH
7.2±n/a
Temperature
310.15±n/a K
IC50
2.5±n/a nM
Comments
extracted
Citation
Naganawa, A; Kusumi, K; Otsuki, K; Sekiguchi, T; Kakuuchi, A; Shinozaki, K; Yamamoto, H; Nonaka, S Phenyl derivative US Patent US8975409 Publication Date 3/10/2015
More Info.:
Target
Name:
Sphingosine 1-phosphate receptor 2
Synonyms:
Edg5 | S1PR2_RAT | S1pr2 | Sphingosine 1-phosphate receptor 2 (S1P2)
Type:
Protein
Mol. Mass.:
38749.58
Organism:
Rattus norvegicus (Rat)
Description:
P47752
Residue:
352
Sequence:
MGGLYSEYLNPEKVQEHYNYTKETLDMQETPSRKVASAFIIILCCAIVVENLLVLIAVARNSKFHSAMYLFLGNLAASDLLAGVAFVANTLLSGPVTLSLTPLQWFAREGSAFITLSASVFSLLAIAIERQVAIAKVKLYGSDKSCRMLMLIGASWLISLILGGLPILGWNCLDHLEACSTVLPLYAKHYVLCVVTIFSVILLAIVALYVRIYFVVRSSHADVAGPQTLALLKTVTIVLGVFIICWLPAFSILLLDSTCPVRACPVLYKAHYFFAFATLNSLLNPVIYTWRSRDLRREVLRPLLCWRQGKGATGRRGGNPGHRLLPLRSSSSLERGLHMPTSPTFLEGNTVV