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Target
Pancreatic alpha-amylase
Ligand
BDBM163655
Substrate
n/a
Meas. Tech.
Kinetic Studies
Temperature
303.15±0 K
Ki
128000±15000 nM
Citation
Williams, LK; Zhang, X; Caner, S; Tysoe, C; Nguyen, NT; Wicki, J; Williams, DE; Coleman, J; McNeill, JH; Yuen, V; Andersen, RJ; Withers, SG; Brayer, GD The amylase inhibitor montbretin A reveals a new glycosidase inhibition motif. Nat Chem Biol 11:691-6 (2015) [PubMed] Article
More Info.:
Target
Name:
Pancreatic alpha-amylase
Synonyms:
1,4-alpha-D-glucan glucanohydrolase | AMY2A | AMYP_HUMAN | PA | Pancreatic α-amylase (HPA) | Pancreatic alpha-amylase | Pancreatic alpha-amylase (HPA)
Type:
Protein
Mol. Mass.:
57709.71
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
511
Sequence:
MKFFLLLFTIGFCWAQYSPNTQQGRTSIVHLFEWRWVDIALECERYLAPKGFGGVQVSPPNENVAIYNPFRPWWERYQPVSYKLCTRSGNEDEFRNMVTRCNNVGVRIYVDAVINHMCGNAVSAGTSSTCGSYFNPGSRDFPAVPYSGWDFNDGKCKTGSGDIENYNDATQVRDCRLTGLLDLALEKDYVRSKIAEYMNHLIDIGVAGFRLDASKHMWPGDIKAILDKLHNLNSNWFPAGSKPFIYQEVIDLGGEPIKSSDYFGNGRVTEFKYGAKLGTVIRKWNGEKMSYLKNWGEGWGFVPSDRALVFVDNHDNQRGHGAGGASILTFWDARLYKMAVGFMLAHPYGFTRVMSSYRWPRQFQNGNDVNDWVGPPNNNGVIKEVTINPDTTCGNDWVCEHRWRQIRNMVIFRNVVDGQPFTNWYDNGSNQVAFGRGNRGFIVFNNDDWSFSLTLQTGLPAGTYCDVISGDKINGNCTGIKIYVSDDGKAHFSISNSAEDPFIAIHAESKL