Reaction Details Report a problem with these data
Target
Mitogen-activated protein kinase 1 [T157A,D319N]
Ligand
BDBM176673
Substrate
n/a
Meas. Tech.
Fluorescence Quenching Assay
Kd
4000±600 nM
Citation
Shapiro, PS; MacKerell, Jr., AD; Fletcher, S Non-ATP dependent inhibitors of extracellular signal-regulated kinase (ERK) US Patent US9115122 Publication Date 8/25/2015
More Info.:
Target
Name:
Mitogen-activated protein kinase 1 [T157A,D319N]
Synonyms:
ERK2(T157A/D319N) | Erk2 | MK01_MOUSE | Mapk | Mapk1 | Prkm1
Type:
n/a
Mol. Mass.:
41248.65
Organism:
Mus musculus (mouse)
Description:
P63085[T157A,D319N]
Residue:
358
Sequence:
MAAAAAAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNATCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSNEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGYRS