Reaction Details Report a problem with these data
Target
Androgen-induced gene 1 protein
Ligand
BDBM195603
Substrate
n/a
Meas. Tech.
Gel-based ABPP Assay
IC50
1.7e+2± 3e+1 nM
Citation
 Parsons, WH; Kolar, MJ; Kamat, SS; Cognetta, AB; Hulce, JJ; Saez, E; Kahn, BB; Saghatelian, A; Cravatt, BF AIG1 and ADTRP are atypical integral membrane hydrolases that degrade bioactive FAHFAs. Nat Chem Biol 12:367-72 (2016) [PubMed]  Article 
Target
Name:
Androgen-induced gene 1 protein
Synonyms:
AIG1 | AIG1_HUMAN | Androgen-induced gene 1 protein (AIG1)
Type:
Protein
Mol. Mass.:
28229.15
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
245
Sequence:
MALVPCQVLRMAILLSYCSILCNYKAIEMPSHQTYGGSWKFLTFIDLVIQAVFFGICVLTDLSSLLTRGSGNQEQERQLKKLISLRDWMLAVLAFPVGVFVVAVFWIIYAYDREMIYPKLLDNFIPGWLNHGMHTTVLPFILIEMRTSHHQYPSRSSGLTAICTFSVGYILWVCWVHHVTGMWVYPFLEHIGPGARIIFFGSTTILMNFLYLLGEVLNNYIWDTQKKPPSWQDMKIKFMYLGPSS
  
Inhibitor
Name:
BDBM195603
Synonyms:
KC01
Type:
Small organic molecule
Emp. Form.:
C22H39NO3
Mol. Mass.:
365.55
SMILES:
CCCCCCCCCCCCCC1OC(=O)\C1=C/CCCCC(N)=O
Structure:
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