Reaction Details Report a problem with these data
Target
Angiopoietin-1 receptor [776-1124]
Ligand
BDBM239657
Substrate
n/a
Meas. Tech.
Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) Assay
pH
7±n/a
Temperature
295.15±n/a K
IC50
0.6±n/a nM
Comments
extracted
Citation
Süβmeier, F; Lobell, M; Grünewald, S; Härter, M; Buchmann, B; Telser, J; Jöriβen, H; Heroult, M; Kahnert, A; Lustig, K; Lindner, N Substituted phenylimidazopyrazoles and their use US Patent US9394309 Publication Date 7/19/2016
More Info.:
Target
Name:
Angiopoietin-1 receptor [776-1124]
Synonyms:
TEK | TIE2 | TIE2_HUMAN | Tyrosine-protein kinase receptor TIE-2 | VMCM | VMCM1
Type:
Enzyme
Mol. Mass.:
39865.58
Organism:
Homo sapiens (Human)
Description:
amino acids 776-1124
Residue:
349
Sequence:
NVQRRMAQAFQNVREEPAVQFNSGTLALNRKVKNNPDPTIYPVLDWNDIKFQDVIGEGNFGQVLKARIKKDGLRMDAAIKRMKEYASKDDHRDFAGELEVLCKLGHHPNIINLLGACEHRGYLYLAIEYAPHGNLLDFLRKSRVLETDPAFAIANSTASTLSSQQLLHFAADVARGMDYLSQKQFIHRDLAARNILVGENYVAKIADFGLSRGQEVYVKKTMGRLPVRWMAIESLNYSVYTTNSDVWSYGVLLWEIVSLGGTPYCGMTCAELYEKLPQGYRLEKPLNCDDEVYDLMRQCWREKPYERPSFAQILVSLNRMLEERKTYVNTTLYEKFTYAGIDCSAEEAA