Assay Method Information

Assay Name:  ChEMBL_1625868 (CHEMBL3868337)
Description:  Antagonist activity at rat OX1 receptor assessed as inhibition of Ala-6,12 orexin-A-induced calcium increase preincubated for 5 mins prior to Ala-6,12 orexin-A addition measured at 1 sec intervals for 1 min by Fluo-4AM dye-based FLIPR assay
Affinity data for this assay
 

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