Assay Method Information

Assay Name:  ChEMBL_1778235 (CHEMBL4235227)
Description:  Antagonist activity at rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced increase in intracellular calcium level pretreated for 5 mins followed by LPC addition by Fluo-4-AM dye based fluorescence assay
Affinity data for this assay
 

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