Compile Data Set for Download or QSAR
maximum 50k data
Found 426 of affinity data for UniProtKB/TrEMBL: O77636
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50227856((3R,4R)-N-hydroxy-4-(4-((2-methylquinolin-4-yl)met...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50227856((3R,4R)-N-hydroxy-4-(4-((2-methylquinolin-4-yl)met...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50183715(CHEMBL207305 | N-(4-(2-(hydroxyamino)-2-oxoethyl)-...)
Affinity DataKi:  0.350nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50183715(CHEMBL207305 | N-(4-(2-(hydroxyamino)-2-oxoethyl)-...)
Affinity DataKi:  0.350nMAssay Description:Inhibition of porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM26526((2R)-N-hydroxy-2-[(3S)-3-methyl-3-{4-[(2-methylqui...)
Affinity DataKi:  0.560nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM26526((2R)-N-hydroxy-2-[(3S)-3-methyl-3-{4-[(2-methylqui...)
Affinity DataKi:  0.560nMAssay Description:Inhibition of porcine TACEMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM26526((2R)-N-hydroxy-2-[(3S)-3-methyl-3-{4-[(2-methylqui...)
Affinity DataKi:  0.560nMAssay Description:Affinity for Tumor necrosis factor alpha converting enzyme (TACE)More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50104974(2,10-Dioxo-11-(2'-trifluoromethyl-biphenyl-4-ylmet...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of porcine TNF-alpha converting enzyme(pTACE).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50104973(2,10-Dioxo-11-(2'-trifluoromethyl-biphenyl-4-ylmet...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of porcine TNF-alpha converting enzyme(pTACE).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50104975((8S,11R,12S)-2,10-Dioxo-11-(2'-trifluoromethyl-bip...)
Affinity DataKi:  2.80nMAssay Description:Inhibition of porcine TNF-alpha converting enzyme(pTACE).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50104977(11-(3',5'-Dichloro-biphenyl-4-ylmethyl)-2,10-dioxo...)
Affinity DataKi:  2.80nMAssay Description:Inhibition of porcine TNF-alpha converting enzyme(pTACE).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50104975((8S,11R,12S)-2,10-Dioxo-11-(2'-trifluoromethyl-bip...)
Affinity DataKi:  2.80nMAssay Description:Inhibition of porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50265114(CHEMBL495502 | N-((2R,6S)-4-(2-(hydroxyamino)-2-ox...)
Affinity DataKi:  2.80nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50104975((8S,11R,12S)-2,10-Dioxo-11-(2'-trifluoromethyl-bip...)
Affinity DataKi:  2.80nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50104978(2,10-Dioxo-11-(3'-trifluoromethyl-biphenyl-4-ylmet...)
Affinity DataKi:  3.70nMAssay Description:Inhibition of porcine TNF-alpha converting enzyme(pTACE).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50104979(2,10-Dioxo-11-(2'-trifluoromethyl-biphenyl-4-ylmet...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of porcine TNF-alpha converting enzyme(pTACE).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50102608(11-Isobutyl-2,10-dioxo-1-oxa-3,9-diaza-cyclopentad...)
Affinity DataKi:  4.20nMAssay Description:Inhibition of porcine TNF-alpha converting enzyme(pTACE).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50102608(11-Isobutyl-2,10-dioxo-1-oxa-3,9-diaza-cyclopentad...)
Affinity DataKi:  4.20nMAssay Description:Inhibition of porcine TNF-alpha converting enzyme (pTACE).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50104976(11-(3',5'-Bis-trifluoromethyl-biphenyl-4-ylmethyl)...)
Affinity DataKi:  4.60nMAssay Description:Inhibition of porcine TNF-alpha converting enzyme(pTACE).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50247674(2-[7-(3,5-Dimethoxy-benzyloxy)-1,1-dioxo-1,3,4,5-t...)
Affinity DataKi:  5nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50104981(11-(2',6'-Difluoro-biphenyl-4-ylmethyl)-2,10-dioxo...)
Affinity DataKi:  6.30nMAssay Description:Inhibition of porcine TNF-alpha converting enzyme(pTACE).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50104980(11-(2'-Methanesulfonyl-biphenyl-4-ylmethyl)-2,10-d...)
Affinity DataKi:  6.5nMAssay Description:Inhibition of porcine TNF-alpha converting enzyme(pTACE).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50102594(7-Isobutyl-8-oxo-2-oxa-9-aza-bicyclo[10.2.2]hexade...)
Affinity DataKi:  12nMAssay Description:Inhibition of porcine TNF-alpha converting enzyme (pTACE).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50136286((3R,4S)-1-(Furan-2-carbonyl)-piperidine-3,4-dicarb...)
Affinity DataIC50:  0.0660nMAssay Description:In vitro binding affinity against porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50229322((3S,4S)-N-hydroxy-4-(4-((2-methylquinolin-4-yl)met...)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50136266((3R,4S)-1-Isobutyryl-piperidine-3,4-dicarboxylic a...)
Affinity DataIC50:  0.220nMAssay Description:In vitro binding affinity against porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50136270((3R,4S)-1-Butyryl-piperidine-3,4-dicarboxylic acid...)
Affinity DataIC50:  0.260nMAssay Description:In vitro binding affinity against porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50136285((3R,4S)-3-Hydroxycarbamoyl-4-[4-(2-methyl-quinolin...)
Affinity DataIC50:  0.280nMAssay Description:In vitro binding affinity against porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50136261((3R,4S)-3-Hydroxycarbamoyl-4-[4-(2-methyl-quinolin...)
Affinity DataIC50: <0.300nMAssay Description:In vitro binding affinity against porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50136283((3R,4S)-1-(Furan-2-carbonyl)-piperidine-3,4-dicarb...)
Affinity DataIC50: <0.300nMAssay Description:In vitro binding affinity against porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50136275((3R,4S)-3-Hydroxycarbamoyl-4-[4-(2-methyl-quinolin...)
Affinity DataIC50: <0.300nMAssay Description:In vitro binding affinity against porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50136262((3R,4S)-1-(1-Methyl-1H-imidazole-4-sulfonyl)-piper...)
Affinity DataIC50:  0.310nMAssay Description:In vitro binding affinity against porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50371344(CHEMBL403401)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50136263((3R,4S)-Piperidine-1,3,4-tricarboxylic acid 1-tert...)
Affinity DataIC50:  0.410nMAssay Description:In vitro binding affinity against porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50136279((3R,4S)-3-Hydroxycarbamoyl-4-[4-(2-methyl-quinolin...)
Affinity DataIC50:  0.440nMAssay Description:In vitro binding affinity against porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50136269((3R,4S)-1-Cyclopropanecarbonyl-piperidine-3,4-dica...)
Affinity DataIC50:  0.450nMAssay Description:In vitro binding affinity against porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50136268((3R,4S)-1-Methanesulfonyl-piperidine-3,4-dicarboxy...)
Affinity DataIC50:  0.480nMAssay Description:In vitro binding affinity against porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50136274((3R,4S)-1-(Furan-2-carbonyl)-piperidine-3,4-dicarb...)
Affinity DataIC50:  0.800nMAssay Description:In vitro binding affinity against porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50136273((3R,4S)-1-Thiazol-2-ylmethyl-piperidine-3,4-dicarb...)
Affinity DataIC50:  0.800nMAssay Description:In vitro binding affinity against porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50152922(CHEMBL184302 | N-Hydroxy-2-{1-[4-(2-methyl-quinoli...)
Affinity DataIC50: <0.800nMAssay Description:Inhibition of porcine Tumor necrosis factor- alpha converting enzyme (TACE, ADAM17)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50136288((3R,4S)-3-Hydroxycarbamoyl-4-[4-(2-methyl-quinolin...)
Affinity DataIC50:  0.830nMAssay Description:In vitro binding affinity against porcine TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50371342(CHEMBL270800)
Affinity DataIC50:  0.940nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50371338(CHEMBL256621)
Affinity DataIC50:  1nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50227849(CHEMBL402746 | CHEMBL537229 | N-((1R,2S)-2-(hydrox...)
Affinity DataIC50:  1nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50371340(CHEMBL271234)
Affinity DataIC50:  1nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50371354(CHEMBL256805)
Affinity DataIC50:  1nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM26808((7S,8R)-7-N-hydroxy-8-N-{4-[(2-methylquinolin-4-yl...)
Affinity DataIC50:  1nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50247718(CHEMBL461801 | N-(3-(hydroxyamino)-3-oxopropyl)-4-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50183725(CHEMBL206254 | N-(4-(2-(hydroxyamino)-2-oxoethyl)-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50129040((((S)-Hydroxycarbamoyl)-{(R)-1-[4-(2-methyl-quinol...)
Affinity DataIC50: <1nMAssay Description:In vitro inhibition of TNF-alpha converting enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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