Compile Data Set for Download or QSAR
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Found 104 of affinity data for UniProtKB/TrEMBL: A2ACE8
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM523902(2-amino-N-[1-(5-chloro-7H-pyrrolo[2,3-d]pyrimidin-...)
Affinity DataIC50:  6.31nMAssay Description:ASK1 and ASK2 biochemical activities were also quantified using AlphaScreen technology which measures the degree of phosphorylation of a protein subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM523902(2-amino-N-[1-(5-chloro-7H-pyrrolo[2,3-d]pyrimidin-...)
Affinity DataIC50:  6.46nMAssay Description:IMAP technology provides a homogeneous assay applicable to a wide variety of kinases, phosphatases, and phosphodiesterases without regard for substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM523865(2-amino-5-methyl-N-[1-(5-methyl-7H-pyrrolo[2,3-d]p...)
Affinity DataIC50:  8.32nMAssay Description:IMAP technology provides a homogeneous assay applicable to a wide variety of kinases, phosphatases, and phosphodiesterases without regard for substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM523862(2-amino-5-fluoro-N-[1-(5-methyl-7H-pyrrolo[2,3-d]p...)
Affinity DataIC50:  11nMAssay Description:IMAP technology provides a homogeneous assay applicable to a wide variety of kinases, phosphatases, and phosphodiesterases without regard for substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM523901(2-amino-5-chloro-N-[1-(5-methyl-7H-pyrrolo[2,3-d]p...)
Affinity DataIC50:  15.8nMAssay Description:ASK1 and ASK2 biochemical activities were also quantified using AlphaScreen technology which measures the degree of phosphorylation of a protein subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM523862(2-amino-5-fluoro-N-[1-(5-methyl-7H-pyrrolo[2,3-d]p...)
Affinity DataIC50:  19.5nMAssay Description:ASK1 and ASK2 biochemical activities were also quantified using AlphaScreen technology which measures the degree of phosphorylation of a protein subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  90.8nMAssay Description:Inhibition of human MEKK6 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50551987(CHEMBL4763562)
Affinity DataIC50:  201nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50552003(CHEMBL4764071)
Affinity DataIC50:  264nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  475nMAssay Description:Inhibition of human MEKK6 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50334268(CHEMBL1642655 | CHEMBL2205637 | N-(6-(1H-imidazol-...)
Affinity DataIC50:  510nMAssay Description:Inhibition of ASK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50551995(CHEMBL4759182)
Affinity DataIC50:  742nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50551972(CHEMBL4776637)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50551992(CHEMBL4751918)
Affinity DataIC50:  1.48E+3nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50551988(CHEMBL4749551)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50551989(CHEMBL4795965)
Affinity DataIC50:  2.34E+3nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50551977(CHEMBL4744931)
Affinity DataIC50:  2.78E+3nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50552004(CHEMBL4753203)
Affinity DataIC50:  2.86E+3nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50551994(CHEMBL4750857)
Affinity DataIC50:  2.91E+3nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50551993(CHEMBL4778358)
Affinity DataIC50:  4.86E+3nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50551998(CHEMBL4740051)
Affinity DataIC50:  4.99E+3nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50552007(CHEMBL4796925)
Affinity DataIC50:  5.29E+3nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50212258(GS-4997 | Selonsertib)
Affinity DataIC50:  6.25E+3nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50552006(CHEMBL4752034)
Affinity DataIC50:  7.17E+3nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50552005(CHEMBL4761865)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ASK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50308060(16-hydroxy-16-(hydroxymethyl)-15-methyl-28-oxa-4,1...)
Affinity DataKd:  170nMAssay Description:Binding affinity to ASK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50326053(CHEMBL608533 | PKC-412)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to ASK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50308060(16-hydroxy-16-(hydroxymethyl)-15-methyl-28-oxa-4,1...)
Affinity DataKd:  170nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50326053(CHEMBL608533 | PKC-412)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50026612(BIBF-1120 | Nintedanib | US10981896, Compound Nint...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataKd:  260nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50300690(1-(5-Tert-Butyl-1,2-Oxazol-3-Yl)-3-(4-{7-[2-(Morph...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to ASK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to ASK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM13535(4-[6-methoxy-7-(3-piperidin-1-ylpropoxy)quinazolin...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to ASK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50326054(CHEMBL1240703)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to ASK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to ASK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM25013(4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3S...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50355495(CHEMBL1908391)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50355496(CHEMBL1908397)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM15138(5-indazolyl pyridine 11g | 5-{5-[(2S)-2-amino-3-ph...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM60665(BDBM50249542 | US9145414, R406 | US9212178, R406)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM27817(2-{[2-({1-[2-(dimethylamino)acetyl]-5-methoxy-2,3-...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50128285(3-(1-Methyl-1H-indol-3-yl)-4-[1-(1-pyridin-2-ylmet...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM50300690(1-(5-Tert-Butyl-1,2-Oxazol-3-Yl)-3-(4-{7-[2-(Morph...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 6(Homo sapiens (Human))
Galapagos

US Patent
LigandPNGBDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ASK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 104 total ) | Next | Last >>
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