Compile Data Set for Download or QSAR
maximum 50k data
Found 290 of affinity data for UniProtKB/TrEMBL: O60755
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187911(1,3-dihydro-1-[3-(2-pyrrolidinylethoxy)phenyl]-3-[...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85168(M32)
Affinity DataKi:  6.03nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85168(M32)
Affinity DataKi:  6.03nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187925(1-(3-(2-(piperidin-1-yl)ethoxy)phenyl)-3-(3-(trifl...)
Affinity DataKi:  8nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85068(Gal(1-13)-Std I)
Affinity DataKi:  8.13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85068(Gal(1-13)-Std I)
Affinity DataKi:  8.13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  9.77nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  9.77nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85200(Galanin (1-19), rat | Galanin rat)
Affinity DataKi:  12.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85200(Galanin (1-19), rat | Galanin rat)
Affinity DataKi:  12.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | GWTLNSAGYLLGPPPGFSPFR-CONH2 | Galan...)
Affinity DataKi:  14.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | GWTLNSAGYLLGPPPGFSPFR-CONH2 | Galan...)
Affinity DataKi:  14.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187919(1-(3-(3-(diethylamino)-2-hydroxypropoxy)phenyl)-3-...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187923(1,3-dihydro-1-phenyl-3-[[3-(trilfluoromethyl)pheny...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187923(1,3-dihydro-1-phenyl-3-[[3-(trilfluoromethyl)pheny...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187922(1-(3-(3-(diethylamino)propoxy)phenyl)-3-(3-(triflu...)
Affinity DataKi:  21nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187912(1-(3-(2-(dimethylamino)ethoxy)phenyl)-3-(3-(triflu...)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187908((S)-1-(3-(3-(diethylamino)-2-hydroxypropoxy)phenyl...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187916(1-(3-(3-(dimethylamino)propoxy)phenyl)-3-(3-(trifl...)
Affinity DataKi:  29nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187918(1-(4-(3-(diethylamino)propoxy)phenyl)-3-(3-(triflu...)
Affinity DataKi:  34nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187914(1-(3-((diethylamino)methoxy)phenyl)-3-(3-(trifluor...)
Affinity DataKi:  38nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85073(CAS_3043476 | Galantide (M15) | NSC_3043476)
Affinity DataKi:  39.8nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85073(CAS_3043476 | Galantide (M15) | NSC_3043476)
Affinity DataKi:  39.8nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187913(1-(3-(4-(diethylamino)butoxy)phenyl)-3-(3-(trifluo...)
Affinity DataKi:  45nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187926(1-(3-(3-(pyrrolidin-1-yl)propoxy)phenyl)-3-(3-(tri...)
Affinity DataKi:  49nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189598(1-(ethylpropyl)-3-{[3-(trifluoromethyl)phenyl]azam...)
Affinity DataKi:  52nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85069(Galanin (2-29), rat | Galanin Porcine 2-29)
Affinity DataKi:  60.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  69.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  69.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187915(1-(4-(4-(diethylamino)butoxy)phenyl)-3-(3-(trifluo...)
Affinity DataKi:  70nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187910(1-(4-(2-(diethylamino)ethoxy)phenyl)-3-(3-(trifluo...)
Affinity DataKi:  78nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187909(1-(3-(2-(diethylamino)ethoxy)phenyl)-3-(3-(trifluo...)
Affinity DataKi:  87nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187917(1-(4-(2-(dimethylamino)ethoxy)phenyl)-3-(3-(triflu...)
Affinity DataKi:  89nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189596(1-(2-propynyl)-3-{[3-(trifluoromethyl)phenyl]azame...)
Affinity DataKi:  89nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189600((E)-1-allyl-3-(3,4-dichlorophenylimino)indolin-2-o...)
Affinity DataKi:  150nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50307254(CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40)
Affinity DataKi:  288nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50307254(CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40)
Affinity DataKi:  288nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187924((R)-1-(3-(3-(diethylamino)-2-hydroxypropoxy)phenyl...)
Affinity DataKi:  290nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50273367((2S,3S)-2-((S)-2-((S)-2-((S)-1-(2-((S)-2-((S)-2-((...)
Affinity DataKi:  316nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50273367((2S,3S)-2-((S)-2-((S)-2-((S)-1-(2-((S)-2-((S)-2-((...)
Affinity DataKi:  316nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189597((E)-3-(2,3-dichlorophenylimino)indolin-2-one | CHE...)
Affinity DataKi:  437nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189595(3-{[3-(trifluoromethyl)phenyl]azamethylene}benzo[d...)
Affinity DataKi:  596nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187920(1-(2-(2-(pyrrolidin-1-yl)ethoxy)phenyl)-3-(3-(trif...)
Affinity DataKi:  790nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189599((E)-3-(4-chlorophenylimino)indolin-2-one | CHEMBL2...)
Affinity DataKi:  850nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85170(Galanin (3-29), porcine)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187921(1-(2-(2-(diethylamino)ethoxy)phenyl)-3-(3-(trifluo...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85170(Galanin (3-29), porcine)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85169(Galanin (1-29), porcine | Galanin [D-Trp2], porcin...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85169(Galanin (1-29), porcine | Galanin [D-Trp2], porcin...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189601((E)-3-(4-methoxyphenylimino)indolin-2-one | (E/Z)-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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