Compile Data Set for Download or QSAR
maximum 50k data
Found 9 for UniProtKB: O88420
TargetSodium channel protein type 8 subunit alpha(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50451447(CHEMBL4217988)
Affinity DataIC50:  5nMAssay Description:Inhibition of rat Nav1.6 expressed in HEK cells by patch clamp electrophysiology methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 8 subunit alpha(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50330763(2-(4-Methoxyphenyl)-4(5)-phenylimidazole | 2-(4-me...)
Affinity DataIC50:  1.96E+4nMAssay Description:Inhibition of rat NaV1.6-mediated current expressed in human HEK293 cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 8 subunit alpha(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50392415(CHEMBL402642)
Affinity DataIC50:  2.85E+4nMAssay Description:Inhibition of rat NaV1.6-mediated current expressed in human HEK293 cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 8 subunit alpha(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50392416(CHEMBL2151778)
Affinity DataIC50:  3.17E+4nMAssay Description:Inhibition of rat NaV1.6-mediated current expressed in human HEK293 cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 8 subunit alpha(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50133778(2,4(5)-Diphenylimidazole | 2,4-diphenyl-1H-imidazo...)
Affinity DataIC50:  3.22E+4nMAssay Description:Inhibition of rat NaV1.6-mediated current expressed in human HEK293 cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 8 subunit alpha(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50392417(CHEMBL2151781)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of rat NaV1.6-mediated current expressed in human HEK293 cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 8 subunit alpha(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50392418(CHEMBL2151783)
Affinity DataIC50:  5.36E+4nMAssay Description:Inhibition of rat NaV1.6-mediated current expressed in human HEK293 cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 8 subunit alpha(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50351882(CHEMBL1825043)
Affinity DataIC50:  1.25E+5nMAssay Description:Inhibition of rat NaV1.6-mediated current expressed in human HEK293 cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3/4/5/8/9/10/11 subunit alpha(Rattus norvegicus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50344821(10-hydroxymethyl-5-imino-(2S)-12,13-dioxa-4,6-diaz...)
Affinity DataKd:  1.80nMAssay Description:Displacement of [3H]saxitoxin from NaV in rat brain membranesMore data for this Ligand-Target Pair