TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 6.80nMAssay Description:Inhibition of mouse uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Inhibition of mouse uPA serine protease domain preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of mouse uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 246nMAssay Description:Inhibition of mouse uPA serine protease domain preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 550nMAssay Description:Inhibition of mouse uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 550nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 550nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 956nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate measured for 15 mins by fluorometric assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 1.61E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 1.77E+3nMAssay Description:Inhibition of mouse uPA serine protease domain preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 2.31E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 2.77E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate measured for 15 mins by fluorometric assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 3.29E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate measured for 15 mins by fluorometric assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 9.31E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.10nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 10nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of uPA in presence of 75% mouse serum measured immediatelyMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of uPA in presence of 75% mouse serum measured at 8 hrsMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of uPA in presence of 75% mouse serum measured at 2 hrsMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Inhibition of uPA in presence of 75% mouse serum measured at 24 hrsMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 79nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 132nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 162nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 644nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 758nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 3.28E+3nMAssay Description:Inhibition of the intrinsic peri-cellular uPA in mouse CT26 cells assessed as reduction in cell invasion measured every hour by transwell assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.02E+3nMAssay Description:Inhibition of the intrinsic peri-cellular uPA in mouse CT26 cells assessed as reduction in cell invasion measured every hour by transwell assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 1.42E+4nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 3.94E+4nMAssay Description:Inhibition of the intrinsic peri-cellular uPA in mouse CT26 cells assessed as reduction in cell invasion measured every hour by transwell assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKd: 11nMAssay Description:Binding affinity to mouse uPA expressed in HEK2936E cells by ITC assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKd: 398nMAssay Description:Binding affinity to mouse uPA by SPR assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKd: 42nMAssay Description:Binding affinity to mouse uPA expressed in HEK2936E cells by ITC assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKd: 15nMAssay Description:Binding affinity to mouse uPA by SPR assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKd: 354nMAssay Description:Binding affinity to mouse uPA expressed in HEK2936E cells by ITC assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKd: 2.40nMAssay Description:Binding affinity to mouse uPA by SPR assayMore data for this Ligand-Target Pair