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Report error Found 166 of affinity data for UniProtKB/TrEMBL: P09884
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50446130(AG-014699 | AG-14447 | Rucaparib | RUCAPARIB CAMSY...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of DNA polymerase alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50231344(CHEMBL334214)
Affinity DataEC50: <1nMAssay Description:Effective concentration against DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50225280(CHEMBL3144215)
Affinity DataKi:  1nMAssay Description:Compound was tested for its inhibitory activity against HeLa DNA polymerase alpha, Ki values were obtained in the absence of dGTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50231343(CHEMBL119038)
Affinity DataEC50: <1nMAssay Description:Effective concentration against DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50231388(CHEMBL119211)
Affinity DataEC50: <1nMAssay Description:Effective concentration against DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50231345(CHEMBL118970)
Affinity DataEC50: <1nMAssay Description:Effective concentration against DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50231384(CHEMBL331025)
Affinity DataEC50: <1nMAssay Description:Effective concentration against DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50231386(CHEMBL331553)
Affinity DataEC50: <1nMAssay Description:Effective concentration against DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50231383(CHEMBL334229)
Affinity DataEC50: <1nMAssay Description:Effective concentration against DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50408427(CHEMBL483492)
Affinity DataIC50: 15nMAssay Description:Compound was evaluated for 50% inhibition of DHBV DNA polymerase (duck hepatitis B virus)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50408426(CHEMBL2092833)
Affinity DataIC50: 480nMAssay Description:Compound was evaluated for 50% inhibition of DHBV DNA polymerase (duck hepatitis B virus)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50443277(CHEMBL5281189)
Affinity DataIC50: 680nMAssay Description:Inhibition of DNA polymerase alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50293303(gallic acid 5,6-dihydroxy-3-carboxyphenylester | C...)
Affinity DataKi:  830nMAssay Description:Inhibition of DNA polymerase alpha from human KB3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50205415(({[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-(5-methyl-2,4-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for 50% inhibition of DHBV DNA polymerase (duck hepatitis B virus)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50042444(6-Methoxy-1,4a-dimethyl-1,2,3,4,4a,9,10,10a-octahy...)
Affinity DataEC50:  1.00E+3nMAssay Description:Effective concentration against DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50205415(({[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-(5-methyl-2,4-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for 50% inhibition of DHBV DNA polymerase (duck hepatitis B virus)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50025592((4-Butyl-phenyl)-(6-methylsulfanyl-9H-purin-2-yl)-...)
Affinity DataKi:  1.00E+3nMAssay Description:Compound was evaluated for the concentration which gives half-maximal inhibition of Chinese Hamster Ovary DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50248359(Adefovir dipivoxil | GS-0840 | Hepsera)
Affinity DataKi:  1.18E+3nMAssay Description:Binding affinity to DNA polymerase alpha (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50025600((4-Butyl-phenyl)-(6-methoxy-9H-purin-2-yl)-amine |...)
Affinity DataKi:  1.40E+3nMAssay Description:Compound was evaluated for the concentration which gives half-maximal inhibition of Chinese Hamster Ovary DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184758((3aS,4S,7R,7aR)-1,6-didodecyl-2,7-bis(methoxycarbo...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184755((3aS,4S,7R,7aR)-1,6-dihexadecyl-2,7-bis(methoxycar...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50090910(6,13-di(hydroxymethyl)-2,6-dimethyl-(1S,2S,5R,6R,7...)
Affinity DataEC50:  2.00E+3nMAssay Description:Effective concentration against DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184757((3aR,4R,7S,7aS)-7-ethyl 2,4-dimethyl 3,5-dihexadec...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50090910(6,13-di(hydroxymethyl)-2,6-dimethyl-(1S,2S,5R,6R,7...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human DNA polymerase alpha using 5' end radiolabeled 24nt DNA/48nt DNA as primer/template after 5 mins by PAGE analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50335554(({[({[2-(2-amino-6-oxo-6,9-dihydro-3H-purin-9-yl)e...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human DNA polymerase alpha by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50090910(6,13-di(hydroxymethyl)-2,6-dimethyl-(1S,2S,5R,6R,7...)
Affinity DataIC50: 2.60E+3nMpH: 7.5Assay Description:Inhibition of human alpha DNA polymerase (95 uL) activity in a solution containg 6.4 mM HEPES (pH 7.5) upon incubation for 12 minutes at 26 degrees C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50025598((4-Butyl-phenyl)-(6-chloro-9H-purin-2-yl)-amine | ...)
Affinity DataKi:  2.60E+3nMAssay Description:Compound was evaluated for the concentration which gives half-maximal inhibition of Chinese Hamster Ovary DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50090910(6,13-di(hydroxymethyl)-2,6-dimethyl-(1S,2S,5R,6R,7...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50090910(6,13-di(hydroxymethyl)-2,6-dimethyl-(1S,2S,5R,6R,7...)
Affinity DataIC50: 3.00E+3nMAssay Description:Compound was evaluated for the inhibitory activity against Human alpha polymeraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50042448(7-Formyl-6-methoxy-1,4a-dimethyl-1,2,3,4,4a,9,10,1...)
Affinity DataEC50:  3.00E+3nMAssay Description:Effective concentration against DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50042456((8-Hydroxymethyl-3-methoxy-4b,8-dimethyl-4b,5,6,7,...)
Affinity DataEC50:  3.00E+3nMAssay Description:Effective concentration against DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM23926(5-[(E)-2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human DNA polymerase-alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184752((3aS,4S,7R,7aR)-1,6-dihexadecyl-2,7-bis(isopropoxy...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184756((3aR,4S,7S,7aS)-7-ethyl 2,4-dimethyl 3,5-dihexadec...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184754((E)-methyl-3,6-dioxo-4-docosenoate | CHEMBL425779)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50153106([(3S,10R,13R,17R)-17-((R)-1,5-Dimethyl-hexyl)-10,1...)
Affinity DataKi:  3.75E+3nMAssay Description:Inhibition constant against DNA polymerase alpha non competitively on dNTP substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50042449(1,7-Bis-hydroxymethyl-1,4a-dimethyl-1,2,3,4,4a,9,1...)
Affinity DataEC50:  4.00E+3nMAssay Description:Effective concentration against DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50042445(6-Methoxy-1,4a-dimethyl-1,2,3,4,4a,9,10,10a-octahy...)
Affinity DataEC50:  4.00E+3nMAssay Description:Effective concentration against DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50090910(6,13-di(hydroxymethyl)-2,6-dimethyl-(1S,2S,5R,6R,7...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human DNA polymerase alpha using 5-end radiolabeled 24nt to 48nt DNA as primer template after 5 mins in presence of dCTP/dGTP/dTTP/dATP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50143526(Untenone A | CHEMBL366792)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50090910(6,13-di(hydroxymethyl)-2,6-dimethyl-(1S,2S,5R,6R,7...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human DNA polymerase alpha using 5-end radiolabeled 24nt to 48nt DNA as primer template after 5 mins in presence of dCTP/dGTP/dTTP/dATP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50042454(7-Formyl-6-hydroxy-1,4a-dimethyl-1,2,3,4,4a,9,10,1...)
Affinity DataEC50:  5.00E+3nMAssay Description:Effective concentration against DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50313784((R)-9-(((2-(benzofuran-2-yl)-2-hydroxyethyl)(methy...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human recombinant DNA polymerase alpha expressed in baculovirus infected SF9 cells after 12 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50313783(N-(4-chlorobenzyl)-1-methyl-9-(morpholinomethyl)-2...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human recombinant DNA polymerase alpha expressed in baculovirus infected SF9 cells after 12 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50025597((4-Butyl-phenyl)-(9H-purin-2-yl)-amine | CHEMBL278...)
Affinity DataKi:  5.00E+3nMAssay Description:Compound was evaluated for the concentration which gives half-maximal inhibition of Chinese Hamster Ovary DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184761((3aR,4R,7S,7aS)-dimethyl 3,5-dihexadecyl-1-oxo-7-(...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50042447(1,7-Bis-hydroxymethyl-1,4a-dimethyl-1,2,3,4,4a,9,1...)
Affinity DataEC50:  7.00E+3nMAssay Description:Effective concentration against DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50013074(2-(4-Butyl-phenylamino)-1,9-dihydro-purin-6-one(Bu...)
Affinity DataKi:  7.50E+3nMAssay Description:Compound was tested for its inhibitory activity against HeLa DNA polymerase alpha, Ki values were obtained in the absence of dGTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50153111([(3S,5S,10S,13R,17R)-17-((R)-1,5-Dimethyl-hexyl)-1...)
Affinity DataKi:  7.84E+3nMAssay Description:Inhibition constant against DNA polymerase alpha non competitively on dNTP substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA polymerase alpha catalytic subunit(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50184750((2R,3S,4R)-4-hydroxy-5-[2-oxo-nonadec-ylidene]-1-p...)
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of DNA polymerase alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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