Compile Data Set for Download or QSAR
Report error Found 2703 of affinity data for UniProtKB/TrEMBL: P17931
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21519(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-(carbam...)
Affinity DataKd:  6.50E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21521(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  3.80E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21522(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  5.20E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21523(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-[(butyl...)
Affinity DataKd:  2.30E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21524(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-[(dieth...)
Affinity DataKd:  4.30E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21525(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  7.40E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21526(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  6.50E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21527(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  4.00E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21528(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-[(benzy...)
Affinity DataKd:  1.50E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21529(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  3.50E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21530(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-[(cyclo...)
Affinity DataKd:  5.70E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21531(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-3,5-dihyd...)
Affinity DataKd:  6.90E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21532(N-[(2R,3R,4R,5S,6R)-5-{[(2S,3R,4S,5R,6R)-4-({[(2S,...)
Affinity DataKd:  1.60E+5nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21533(N-[(2R,3R,4R,5S,6R)-4-hydroxy-6-(hydroxymethyl)-2-...)
Affinity DataKd:  6.70E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21534([(2S,3R,4S,5R,6R)-5-hydroxy-6-(hydroxymethyl)-4-[(...)
Affinity DataKd:  8.70E+4nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21535({[(2S,3R,4S,5R,6R)-5-hydroxy-6-(hydroxymethyl)-4-[...)
Affinity DataKd:  1.50E+5nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21536({[(2S,3R,4S,5R,6R)-5-hydroxy-6-(hydroxymethyl)-4-[...)
Affinity DataKd:  2.50E+5nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21537((benzyloxy)({[(2S,3R,4S,5R,6R)-5-hydroxy-6-(hydrox...)
Affinity DataKd:  1.20E+5nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21538((2S,3R,4S,5R,6R)-5-hydroxy-6-(hydroxymethyl)-4-[(4...)
Affinity DataKd:  2.40E+5nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21539(N-[(2S,3R,4S,5R,6R)-3-(benzyloxy)-5-hydroxy-6-(hyd...)
Affinity DataKd:  3.80E+5nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21540(N-[(2R,3R,4S,5R,6S)-3,5-dihydroxy-2-(hydroxymethyl...)
Affinity DataKd:  2.20E+5nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21541((2R,3R,4S,5R,6S)-2-(hydroxymethyl)-6-(methylsulfan...)
Affinity DataKd:  5.90E+6nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM21542([(2S,3R,4S,5R,6R)-4,5-dihydroxy-6-(hydroxymethyl)-...)
Affinity DataKd:  2.80E+6nMpH: 7.2 T: 2°CAssay Description:In fluorescence polarization measurements, a fluorescent probe was excited with plane-polarized light and the degree of polarization remaining in the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2008
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM120768(US8703720, Reference Compound 1)
Affinity DataKd:  4.40E+6nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM120769(US8703720, Reference Compound 2)
Affinity DataKd:  5.90E+4nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM120770(US8703720, 7)
Affinity DataKd:  430nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM120771(US8703720, 15)
Affinity DataKd:  230nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM120772(US8703720, 16)
Affinity DataKd:  150nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM120773(US8703720, 17)
Affinity DataKd:  210nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM120774(US8703720, 18)
Affinity DataKd:  550nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM120775(US8703720, 19)
Affinity DataKd:  190nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM120776(US8703720, 23)
Affinity DataKd:  1.40E+3nMAssay Description:Compounds 7, 15-19, and 22 were evaluated for their efficiency in inhibiting galectin-1 and galectin-3 in a known fluorescence polarization-based ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2014
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM223990(2-[6-Maleimide)caproyl]ethyl [3-O-(2-naphthyl)meth...)
Affinity DataKd:  14nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2017
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM223990(2-[6-Maleimide)caproyl]ethyl [3-O-(2-naphthyl)meth...)
Affinity DataKd:  82nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2017
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM223991([3-O-(2-naphthyl)methyl-β-D-galactopyranosyl]...)
Affinity DataKd:  590nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2017
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM223991([3-O-(2-naphthyl)methyl-β-D-galactopyranosyl]...)
Affinity DataKd:  2.99E+3nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2017
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM223992(4-O-[3-O-(3-methoxybenzyl)-β-D-galactopyranos...)
Affinity DataKd:  660nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2017
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM223992(4-O-[3-O-(3-methoxybenzyl)-β-D-galactopyranos...)
Affinity DataKd:  3.27E+3nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2017
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM223993(TD139)
Affinity DataKd:  36nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2017
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM223993(TD139)
Affinity DataKd:  166nMT: 2°CAssay Description:Fluorescence anisotropy was measured on a Tecan infinite M1000 plate reader with an excitation at 470 nm and emission at 525 nm, using Greiner 96 fla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2017
Entry Details Article
PubMed
TargetGalectin-3(Human)
Lund University

LigandPNGBDBM455401(3,3'-Dideoxy-3- [4-(morpholin-4- yl)-1H-1,2,3- tri...)
Affinity DataKd:  2nMAssay Description:The affinity of Example 1-5 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the inter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM455402(3,3′-Dideoxy-3-[4-(4-methylpiperazin-1-yl)-1...)
Affinity DataKd:  7nMAssay Description:The affinity of Example 1-5 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the inter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM455403(3,3′-Dideoxy-3-[4-(piperidin-4-yl)-1H-1,2,3-...)
Affinity DataKd:  5nMAssay Description:The affinity of Example 1-5 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the inter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM455404(3,3′-Dideoxy-3-[4-(tetrahydropyran-4-yl)-1H-...)
Affinity DataKd:  1nMAssay Description:The affinity of Example 1-5 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the inter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM455405(3,3′-Dideoxy-3-[4-(propan-2-yl)-1H-1,2,3-tri...)
Affinity DataKd:  2nMAssay Description:The affinity of Example 1-5 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the inter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM461806(3,4-Dimethylphenyl 3-deoxy-3-[4-(3,4,5-triflooroph...)
Affinity DataKd:  150nMAssay Description:The affinity of Example 1-106 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the int...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2021
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM461807(3-Bromophenyl 3-deoxy-3-[4-(3,4,5-trifluorophenyl)...)
Affinity DataKd:  37nMAssay Description:The affinity of Example 1-106 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the int...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2021
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM461808(3-Ethoxyphenyl 3-deoxy-3-[4-(3,4,5-trifluorophenyl...)
Affinity DataKd:  420nMAssay Description:The affinity of Example 1-106 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the int...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2021
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM461809(4-Pyridyl 3-deoxy-1-thio-3-[4-(3,4,5-trifluorophen...)
Affinity DataKd:  190nMAssay Description:The affinity of Example 1-106 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the int...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2021
Entry Details
Go to US Patent

TargetGalectin-3(Human)
Lund University

LigandPNGBDBM461810(2,4-Dichlorophenyl 3-deoxy-3-[4-(3,4,5-trifluoroph...)
Affinity DataKd:  650nMAssay Description:The affinity of Example 1-106 for galectins were determined by a fluorescence anisotropy assay where the compound was used as an inhibitor of the int...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2021
Entry Details
Go to US Patent

Displayed 1 to 50 (of 2703 total ) | Next | Last >>
Jump to: