Compile Data Set for Download or QSAR
Report error Found 271 for UniProtKB: P22002
LigandChemical structure of BindingDB Monomer ID 50336640BDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataKi:  0.130nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50318494BDBM50318494(3-ethyl 5-methyl 2,6-dimethyl-4-(3-nitrophenyl)-1,...)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50336640BDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 82056BDBM82056(CAS_4499 | NSC_4499 | Nisoldipine)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50318494BDBM50318494(3-ethyl 5-methyl 2,6-dimethyl-4-(3-nitrophenyl)-1,...)
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 82056BDBM82056(CAS_4499 | NSC_4499 | Nisoldipine)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50318493BDBM50318493(Nimotop | 3-isopropyl 5-(2-methoxyethyl) 2,6-dimet...)
Affinity DataKi:  0.560nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50336640BDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50318493BDBM50318493(Nimotop | 3-isopropyl 5-(2-methoxyethyl) 2,6-dimet...)
Affinity DataKi:  0.790nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50336640BDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of rat Cav1.2 channel in rat mesenteric artery assessed as relaxation of 70 mM K+ induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50318494BDBM50318494(3-ethyl 5-methyl 2,6-dimethyl-4-(3-nitrophenyl)-1,...)
Affinity DataKi:  1.76nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2011
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 79180BDBM79180(MLS001331726 | cid_60496 | benzenesulfonic acid;3-...)
Affinity DataKi:  2nMAssay Description:Binding affinity against rat L-type calcium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50336640BDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataKi:  2.06nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2011
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50079458BDBM50079458(2,6-Dimethyl-4-[3-methyl-5-(2-naphthalen-1-yl-ethy...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50231571BDBM50231571(CHEMBL3350845)
Affinity DataKi:  2.20nMAssay Description:Inhibition of [3H](+)-PN200-110 binding to L-type calcium channel 1,4-DHP binding site of rat ventricular myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50318493BDBM50318493(Nimotop | 3-isopropyl 5-(2-methoxyethyl) 2,6-dimet...)
Affinity DataKi:  2.28nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2011
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50231574BDBM50231574(CHEMBL3350842)
Affinity DataKi:  2.40nMAssay Description:Inhibition of [3H](+)-PN200-110 binding to L-type calcium channel 1,4-DHP binding site of rat ventricular myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 82057BDBM82057(NSC_65832 | NSC_107928 | CAS_65832 | D888,(+) | CA...)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2011
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 82056BDBM82056(CAS_4499 | NSC_4499 | Nisoldipine)
Affinity DataKi:  2.79nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2011
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50336640BDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of [3H](+)-PN200-110 binding to L-type calcium channel 1,4-DHP binding site of rat ventricular myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50453799BDBM50453799(Niguldipine)
Affinity DataKi:  4.60nMAssay Description:Binding affinity for rat L-type [Ca2+] channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50079463BDBM50079463(4-{5-[2-(3-Bromo-phenyl)-ethyl]-3-phenyl-isoxazol-...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 26948BDBM26948(CHEMBL46516 | cid_3396 | FLUSPIRILENE | 8-[4,4-bis...)
Affinity DataKi:  7.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50029426BDBM50029426([2-(3,4-Dimethoxy-phenyl)-ethyl]-[4-(4-methoxy-phe...)
Affinity DataKi:  8.30nMAssay Description:Calcium antagonistic activity by measuring [3H]nitrendipine displacement from rat heart L-type [Ca2+] channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50079459BDBM50079459(4-[5-(2-Biphenyl-4-yl-ethyl)-3-methyl-isoxazol-4-y...)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50453799BDBM50453799(Niguldipine)
Affinity DataKi:  9nMAssay Description:Inhibition of [3H]nitrendipine binding to membrane homogenates of of rat cardiac muscle.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 82057BDBM82057(NSC_65832 | NSC_107928 | CAS_65832 | D888,(+) | CA...)
Affinity DataKi:  9.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2011
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50030617BDBM50030617(2,6-Dimethyl-4-(4-nitro-phenyl)-pyridine-3,5-dicar...)
Affinity DataKi: >10nMAssay Description:Inhibition of [3H]nitrendipine binding to membrane homogenates of of rat cardiac muscle.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 81939BDBM81939(NSC_62969 | VERAPAMIL | CAS_52-53-9)
Affinity DataKi:  10.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50079464BDBM50079464(2,6-Dimethyl-4-[3-methyl-5-(2-naphthalen-2-yl-ethy...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50052311BDBM50052311(Acetic acid (4R,5R)-7-chloro-1-dimethylaminomethyl...)
Affinity DataIC50: 12nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50231573BDBM50231573(CHEMBL3350846)
Affinity DataKi:  14nMAssay Description:Inhibition of [3H](+)-PN200-110 binding to L-type calcium channel 1,4-DHP binding site of rat ventricular myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50231570BDBM50231570(CHEMBL3350843)
Affinity DataKi:  16nMAssay Description:Inhibition of [3H](+)-PN200-110 binding to L-type calcium channel 1,4-DHP binding site of rat ventricular myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50231572BDBM50231572(CHEMBL3350844)
Affinity DataKi:  17nMAssay Description:Inhibition of [3H](+)-PN200-110 binding to L-type calcium channel 1,4-DHP binding site of rat ventricular myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50042750BDBM50042750({8-[5-Methoxycarbonyl-2,6-dimethyl-4-(2-trifluorom...)
Affinity DataKi:  17nMAssay Description:Inhibition of [3H](+)-PN200-110 binding to L-type calcium channel 1,4-DHP binding site of rat ventricular myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50029417BDBM50029417([4-(4-Methoxy-phenyl)-4H-benzo[b]pyrrolo[1,2-d][1,...)
Affinity DataIC50: 17nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50042752BDBM50042752({12-[5-Methoxycarbonyl-2,6-dimethyl-4-(2-trifluoro...)
Affinity DataKi:  17nMAssay Description:Inhibition of [3H](+)-PN200-110 binding to L-type calcium channel 1,4-DHP binding site of rat ventricular myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 82061BDBM82061(GALLOPAMIL | CAS_119442 | NSC_119442 | D600)
Affinity DataKi:  21.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2011
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50101905BDBM50101905(Fantofarone | SR-33557)
Affinity DataIC50: 22nMAssay Description:Inhibition of L-type calcium channel measured using whole-cell patch clamp in rat ventricular myocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2016
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 82061BDBM82061(GALLOPAMIL | CAS_119442 | NSC_119442 | D600)
Affinity DataKi:  22.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2011
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50079462BDBM50079462(2,6-Dimethyl-4-(3-methyl-5-phenethyl-isoxazol-4-yl...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50029415BDBM50029415((6-Chloro-4,4-diphenyl-4H-benzo[b]pyrrolo[1,2-d][1...)
Affinity DataKi:  26nMAssay Description:Calcium antagonistic activity by measuring [3H]nitrendipine displacement from rat heart L-type [Ca2+] channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50030621BDBM50030621(5-[3-(4,4-Diphenyl-piperidin-1-yl)-propylcarbamoyl...)
Affinity DataKi:  30nMAssay Description:Inhibition of [3H]nitrendipine binding to membrane homogenates of of rat cardiac muscle.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50079460BDBM50079460(4-{5-[2-(3-Methoxy-phenyl)-ethyl]-3-phenyl-isoxazo...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50283421BDBM50283421(((E)-Azacyclotridec-1-en-2-yl)-(2,2-diphenyl-penty...)
Affinity DataEC50:  34nMAssay Description:Binding of [3H]nitrendipine to calcium channel in rat heart membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50029424BDBM50029424((3aR,4R)-4-(4-Methoxy-phenyl)-2,3,3a,4-tetrahydro-...)
Affinity DataKi:  35nMAssay Description:Calcium antagonistic activity by measuring [3H]nitrendipine displacement from rat heart L-type [Ca2+] channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 81939BDBM81939(NSC_62969 | VERAPAMIL | CAS_52-53-9)
Affinity DataKi:  38nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 81939BDBM81939(NSC_62969 | VERAPAMIL | CAS_52-53-9)
Affinity DataIC50: 39nMAssay Description:Ability to inhibit [3H]nitrendipine binding to the L-type calcium channel receptor(CCR) in rat heart homogenate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50026636BDBM50026636(RAUWOLSCINE HYDROCHLORIDE | 17alpha-hydroxy-20alph...)
Affinity DataKi:  40nMAssay Description:Inhibition of [3H]nitrendipine binding to membrane homogenates of rat cardiac muscle.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 81939BDBM81939(NSC_62969 | VERAPAMIL | CAS_52-53-9)
Affinity DataKi:  40.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2011
Entry Details
PubMed
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