Compile Data Set for Download or QSAR
Report error Found 85 for UniProtKB: P22007
LigandChemical structure of BindingDB Monomer ID 50080764BDBM50080764((S)-2-({5-[(Benzyl-pyridin-3-yl-amino)-methyl]-2'-...)
Affinity DataIC50: 0.100nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50067563BDBM50067563((S)-2-{[2'-Methyl-5-(pyridin-3-yloxymethyl)-biphen...)
Affinity DataIC50: 0.400nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50067584BDBM50067584(2-{[5-((R)-2-Amino-3-mercapto-propylamino)-bipheny...)
Affinity DataIC50: 0.780nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50072626BDBM50072626(2-[2-({2-[2-(4-Cyano-benzylsulfanyl)-acetylamino]-...)
Affinity DataIC50: 5.40nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50104054BDBM50104054(4-Methylsulfanyl-2-{[5-(5-phenyl-furan-2-ylmethoxy...)
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50104052BDBM50104052(2-{2-[(2-{2-[1-(4-Cyano-benzyl)-4,5-dihydro-1H-imi...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50104047BDBM50104047(N-[3-Benzoyl-4-(2-p-tolyl-acetylamino)-phenyl]-3-[...)
Affinity DataIC50: 35nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103281BDBM50103281(1-(3-Benzoyl-4-diphenylacetylamino-phenylcarbamoyl...)
Affinity DataIC50: 36nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50366477BDBM50366477(CHEMBL69330)
Affinity DataKd:  75nMAssay Description:Inhibition of yeast Farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50103269BDBM50103269(1-{3-Benzoyl-4-[2-(4-bromo-phenyl)-acetylamino]-ph...)
Affinity DataIC50: 76nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103285BDBM50103285(1-[3-Benzoyl-4-(2-p-tolyl-acetylamino)-phenylcarba...)
Affinity DataIC50: 77nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103271BDBM50103271(1-(3-Benzoyl-4-phenylmethanesulfonylamino-phenylca...)
Affinity DataIC50: 85nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 238364BDBM238364(3-(4-(Methoxycarbonyl)phenyl)-4-cyano-5-(isopropyl...)
Affinity DataIC50: 85nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103280BDBM50103280(1-(3-Benzoyl-4-p-tolylmethanesulfonylamino-phenylc...)
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103262BDBM50103262(1-{3-Benzoyl-4-[2-(4-chloro-phenyl)-acetylamino]-p...)
Affinity DataIC50: 105nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 238353BDBM238353(3-(4-Chlorophenyl)-4-cyano-5-(isopropylthio)thioph...)
Affinity DataIC50: 110nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103274BDBM50103274(1-{3-Benzoyl-4-[2-(4-nitro-phenyl)-acetylamino]-ph...)
Affinity DataIC50: 115nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103261BDBM50103261(1-{3-Benzoyl-4-[2-(2,4-dichloro-phenyl)-acetylamin...)
Affinity DataIC50: 120nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 238367BDBM238367(3-(4-Tolyl)-4-cyano-5-(isopropylthio)thiophene-2-c...)
Affinity DataIC50: 190nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 238361BDBM238361(3-(4-Methoxyphenyl)-4-cyano-5-(isopropylthio)thiop...)
Affinity DataIC50: 250nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 238356BDBM238356(3-(4-Fluorophenyl)-4-cyano-5-(isopropylthio)thioph...)
Affinity DataIC50: 270nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 238371BDBM238371(3-(2-Naphthyl)-4-cyano-5-(isopropylthio)thiophene-...)
Affinity DataIC50: 320nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103270BDBM50103270(1-{3-Benzoyl-4-[2-(2,6-dichloro-phenyl)-acetylamin...)
Affinity DataIC50: 340nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 238374BDBM238374(3-(3-Thienyl)-4-cyano-5-(isopropylthio)thiophene-2...)
Affinity DataIC50: 350nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103272BDBM50103272(1-[3-Benzoyl-4-(2-naphthalen-1-yl-acetylamino)-phe...)
Affinity DataIC50: 380nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50289981BDBM50289981({[(2E,6E)-8-[(3-benzoylphenyl)carbonyloxy]-3,7-dim...)
Affinity DataKi:  380nMAssay Description:Inhibition of yeast Farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50104050BDBM50104050(5-Phenyl-pentanoic acid [3-benzoyl-4-(2-p-tolyl-ac...)
Affinity DataIC50: 390nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103260BDBM50103260(1-[3-Benzoyl-4-(2-o-tolyl-acetylamino)-phenylcarba...)
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103258BDBM50103258(1-{3-Benzoyl-4-[2-(2,3-dichloro-phenyl)-acetylamin...)
Affinity DataIC50: 420nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50104055BDBM50104055(N-[3-Benzoyl-4-(2-p-tolyl-acetylamino)-phenyl]-3-[...)
Affinity DataIC50: 455nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 238357BDBM238357(3-(3-Fluorophenyl)-4-cyano-5-(isopropylthio)thioph...)
Affinity DataIC50: 460nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103277BDBM50103277(1-[3-Benzoyl-4-(2-naphthalen-2-yl-acetylamino)-phe...)
Affinity DataIC50: 460nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103284BDBM50103284(1-{3-Benzoyl-4-[2-(3,4-dichloro-phenyl)-acetylamin...)
Affinity DataIC50: 480nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50104048BDBM50104048(N-[3-Benzoyl-4-(2-p-tolyl-acetylamino)-phenyl]-4-p...)
Affinity DataIC50: 530nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103276BDBM50103276(1-{3-Benzoyl-4-[2-(3,5-dichloro-phenyl)-acetylamin...)
Affinity DataIC50: 535nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103259BDBM50103259(1-[3-Benzoyl-4-(2-m-tolyl-acetylamino)-phenylcarba...)
Affinity DataIC50: 540nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103268BDBM50103268(1-{3-Benzoyl-4-[2-(4-methoxy-phenyl)-acetylamino]-...)
Affinity DataIC50: 545nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103257BDBM50103257(1-[3-Benzoyl-4-(4-carboxy-butyrylamino)-phenylcarb...)
Affinity DataIC50: 550nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 238359BDBM238359(3-(4-(Trifluoromethyl)phenyl)-4-cyano-5-(isopropyl...)
Affinity DataIC50: 580nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 238366BDBM238366(3-Phenyl-4-cyano-5-(isopropylthio)thiophene-2-carb...)
Affinity DataIC50: 610nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 238365BDBM238365(3-(3-(Methoxycarbonyl)phenyl)-4-cyano-5-(isopropyl...)
Affinity DataIC50: 620nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 238373BDBM238373(3-(3-Biphenyl)-4-cyano-5-(isopropylthio)thiophene-...)
Affinity DataIC50: 640nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103287BDBM50103287(1-(3-Benzoyl-4-phenylacetylamino-phenylcarbamoyl)-...)
Affinity DataIC50: 650nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103278BDBM50103278(1-[3-Benzoyl-4-(2-phenyl-propionylamino)-phenylcar...)
Affinity DataIC50: 650nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50103266BDBM50103266(1-[3-Benzoyl-4-(3-carboxy-propionylamino)-phenylca...)
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50289982BDBM50289982(Prenyl pyrophosphate analogue)
Affinity DataKi:  700nMAssay Description:Inhibition of yeast Farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50103283BDBM50103283(1-{3-Benzoyl-4-[2-(4-trifluoromethyl-phenyl)-acety...)
Affinity DataIC50: 725nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50104053BDBM50104053(N-[3-Benzoyl-4-(2-p-tolyl-acetylamino)-phenyl]-3-[...)
Affinity DataIC50: 925nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50289979BDBM50289979({[(2E)-4-[(3-benzoylphenyl)carbonyloxy]-3-methylbu...)
Affinity DataKi:  960nMAssay Description:Inhibition of yeast Farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 238375BDBM238375(3-(1-Dibenzofuranyl)-4-cyano-5-(isopropylthio)thio...)
Affinity DataIC50: 1.00E+3nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details Article
PubMed
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