TargetType-1 angiotensin II receptor B(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: >0.000100nMAssay Description:Compound was evaluated for its binding affinity towards rat Angiotensin II receptor, type 1More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor B(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 0.126nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor B(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 0.160nMpH: 7.4Assay Description:Binding affinity for angiotensin II receptor, type 1 in rat liver membrane using [125I]-Ang II as radioligand, in pH 7.4 Tris-HCl buffer for 2 hr at ...More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:In vitro binding affinity against Angiotensin II receptor, type 1 from rat liver membranesMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor B(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
TargetType-1 angiotensin II receptor B(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 0.230nMAssay Description:In vitro binding affinity at rat liver Angiotensin II receptor, type 1 was determined based on displacement of [125I]-Ang IIMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 0.316nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 0.398nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 0.398nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity of compound in presence of bovine serum albumin (BSA) at 0% against rat adrenal Angiotensin II receptor, type 1More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 0.501nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Affinity DataKi: 0.530nMAssay Description:In vitro binding affinity against Angiotensin II receptor, type 1 from rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity towards Angiotensin II receptor, type 1 in rat aortic smooth muscle cells using 0.2 nM [125I]-labeled Sar-Ile-angiotensin IIMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding against Angiotensin II receptor in a radioligand binding assay using [125I]-Sar1-Ile8 angiotensin-II as radioligand in rat adrenal cortical m...More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor B(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 0.619nMAssay Description:Inhibition of binding of [125I]All at the angiotensin II type 1 receptor (AT1 receptor) in rat liver membranesMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 0.631nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor B(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 0.740nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor B(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 0.760nMAssay Description:Compound was evaluated for binding affinity against angiotensin II receptor, type 1 in rat liverMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 0.794nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 0.794nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor B(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 determined using [125I]- labeled [Sar1,Ile8] angiotensin II in rat adrenocortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding against Angiotensin II receptor in a radioligand binding assay using [125I]-Sar1-Ile8 angiotensin-II as radioligand in rat adrenal cortical m...More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor B(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Compound was evaluated for its binding affinity towards rat Angiotensin II receptor, type 1More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 0.850nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor B(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
TargetType-1 angiotensin II receptor B(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition of [125I]- Sar,Ile8-angiotensin II binding to rat adrenal corticcal membrane angiotensin II receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor B(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [125I]-Sar1-Ile8-A II from rat adrenal Angiotensin-1 (AT-1) receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor B(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Inhibition of [125I]- Sar,Ile8-angiotensin II binding to rat adrenal corticcal membrane angiotensin II receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity of compound in presence of bovine serum albumin (BSA) at 0.01% against rat adrenal Angiotensin II receptor, type 1More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity towards Angiotensin II receptor, type 1 in rat aortic smooth muscle cells using 0.2 nM [125I]-labeled Sar-Ile-angiotensin IIMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Glaxo Research And Development
Curated by ChEMBL
Glaxo Research And Development
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair