Compile Data Set for Download or QSAR
maximum 50k data
Found 35 of affinity data for UniProtKB/TrEMBL: P35383
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50118213(5'-UTP | CHEMBL336296 | H4utp | UTP | uridine 5'-(...)
Affinity DataIC50:  1.51E+3nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50029031(1-Amino-4-{4-[4-chloro-6-(3-sulfo-phenylamino)-[1,...)
Affinity DataIC50:  5.00E+3nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336792(CHEMBL256688 | sodium 1-amino-4-(2,4-dimethylpheny...)
Affinity DataIC50:  9.00E+3nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336767(CHEMBL257495 | PSB-716 | sodium 1-amino-4-(2-metho...)
Affinity DataIC50:  9.00E+3nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50371701(CHEMBL271881)
Affinity DataIC50:  9.00E+3nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336786(CHEMBL256864 | sodium 1-amino-9,10-dioxo-4-(o-toly...)
Affinity DataIC50:  1.00E+4nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50227032(CHEMBL256057 | acid blue 25 | sodium 1-amino-9,10-...)
Affinity DataIC50:  1.11E+4nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50227015(CHEMBL271688 | Sodium 1-amino-4-(4-acetylaminophen...)
Affinity DataIC50:  1.20E+4nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336791(CHEMBL402239 | sodium 1-amino-4-(2,3-dimethylpheny...)
Affinity DataIC50:  1.40E+4nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50371703(CHEMBL256689)
Affinity DataIC50:  1.70E+4nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50227023(1-amino-4-(4-methoxyphenyl)-2-sulfoanthraquinone |...)
Affinity DataIC50:  1.70E+4nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336769(CHEMBL403051 | sodium 1-amino-4-(2-ethoxyphenylami...)
Affinity DataIC50:  1.70E+4nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50227019(CHEMBL271673 | sodium 1-amino-4-(4-chlorophenylami...)
Affinity DataIC50:  2.00E+4nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336787(CHEMBL445413 | sodium 1-amino-9,10-dioxo-4-(m-toly...)
Affinity DataIC50:  2.20E+4nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50371702(CHEMBL402238)
Affinity DataIC50:  2.40E+4nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336788(CHEMBL404450 | sodium 1-amino-9,10-dioxo-4-(p-toly...)
Affinity DataIC50:  2.70E+4nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50227016(CHEMBL401859 | Sodium 1-amino-4-(4-anilinophenylam...)
Affinity DataIC50:  3.00E+4nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50378134(CHEMBL572657)
Affinity DataIC50:  9.20E+4nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50371704(CHEMBL270415)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50227018(CHEMBL404659 | Sodium 1-amino-4-(3-nitrophenylamin...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50227020(CHEMBL271672 | sodium 1-amino-4-(3-chlorophenylami...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50371700(CHEMBL271689)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor in mouse NG108-15 cells assessed as inhibition of UTP-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50378133(CHEMBL584184)
Affinity DataIC50:  1.66E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50378128(CHEMBL575653)
Affinity DataIC50:  2.64E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50378126(CHEMBL572422)
Affinity DataIC50:  2.67E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50378130(CHEMBL574076)
Affinity DataIC50:  3.38E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50378132(CHEMBL574529)
Affinity DataIC50:  5.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50378131(CHEMBL575202)
Affinity DataIC50: >5.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50378129(CHEMBL575649)
Affinity DataIC50:  5.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50378127(CHEMBL574998)
Affinity DataIC50: >5.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50378124(CHEMBL572897)
Affinity DataIC50:  5.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50378123(CHEMBL582936)
Affinity DataIC50:  5.00E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 1 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50378125(CHEMBL572655)
Affinity DataIC50:  5.96E+5nMAssay Description:Antagonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as inhibition of 3 uM UTP-induced intracellular calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50378595(CHEMBL605786)
Affinity DataEC50:  9.90E+4nMAssay Description:Agonist activity at mouse P2Y2 receptor expressed in human 1321N1 cells assessed as calcium elevation by fura2/AM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50118213(5'-UTP | CHEMBL336296 | H4utp | UTP | uridine 5'-(...)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at mouse P2Y2 receptor expressed in NG108-15 hybrid cells assessed as increase in intracellular calcium release by fluorescence assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed