TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: >4.00E+4nMAssay Description:Inhibition of human p97 in human HeLa cells harboring UbG76V-GFP assessed as accumulation of UbG76V after 6 hrs by microscopic analysisMore data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 1.90E+4nMAssay Description:Inhibition of human p97 in human HeLa cells harboring UbG76V-GFP assessed as accumulation of UbG76V after 1 hr by microscopic analysisMore data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Inhibition of human p97 in human HeLa cells harboring UbG76V-GFP assessed as accumulation of UbG76V after 6 hrs by microscopic analysisMore data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 1.40E+3nMAssay Description:Inhibition of human p97 in human HeLa cells harboring UbG76V-GFP assessed as accumulation of UbG76V after 1 hr by microscopic analysisMore data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 1.50E+4nMAssay Description:Inhibition of human p97 in human HeLa cells harboring UbG76V-GFP assessed as accumulation of UbG76V after 1 hr by microscopic analysisMore data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: >4.00E+4nMAssay Description:Inhibition of human p97 in human HeLa cells harboring UbG76V-GFP assessed as accumulation of UbG76V after 6 hrs by microscopic analysisMore data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataKd: 5.00E+3nMAssay Description:Binding affinity to p97 (unknown origin) by SPR assayMore data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataKd: 7.00E+3nMAssay Description:Binding affinity to GST-tagged p97 (unknown origin) by CD spectroscopyMore data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: >4.00E+4nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 940nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 1.80E+3nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 2.40E+3nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 2.50E+3nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: >4.00E+4nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 4.70E+4nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: >4.00E+4nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: >4.00E+4nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 4.50E+3nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 1.90E+3nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 2.70E+3nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 2.70E+3nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: >4.00E+4nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 1.10E+4nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 1.30E+3nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 890nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 820nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 1.80E+3nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 820nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 360nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 360nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 1.30E+3nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 640nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 230nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 2.70E+3nMAssay Description:Inhibition of p97 in human HeLa cells expressing UbG76V-GFP/ODD-Luc assessed as accumulation of Ub-GFP incubated for 6 hrs by confocal microscopic an...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 520nMAssay Description:Inhibition of VCP in human HeLa cells assessed as stabilization of ubiquitin-tagged luciferase after 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 90nMAssay Description:Inhibition of VCP in human HeLa cells assessed as stabilization of ubiquitin-tagged luciferase after 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataEC50: 200nMAssay Description:Inhibition of VCP in human HeLa cells assessed as stabilization of ubiquitin-tagged luciferase after 24 hrs by reporter gene assayMore data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:Covalent inhibition of p97 (unknown origin) ATPase activity incubated for 60 mins in presence of ATP by Biomol Green Reagent based microplate reader ...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataIC50: 0.360nMAssay Description:Covalent inhibition of p97 (unknown origin) ATPase activity incubated for 60 mins in presence of ATP by Biomol Green Reagent based microplate reader ...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Covalent inhibition of p97 (unknown origin) ATPase activity incubated for 60 mins in presence of ATP by Biomol Green Reagent based microplate reader ...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataIC50: 3.70nMAssay Description:Covalent inhibition of p97 (unknown origin) ATPase activity incubated for 60 mins in presence of ATP by Biomol Green Reagent based microplate reader ...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Covalent inhibition of p97 (unknown origin) ATPase activity incubated for 60 mins in presence of ATP by Biomol Green Reagent based microplate reader ...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of human p97 ATPase incubated for 15 mins by ADP Glo luminescence assayMore data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Biomol Green (Enzo) is a bioluminescent, homogeneous assay that measures ADP formed from a biochemical reaction. Because of its high sensitivity, the...More data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of p97 (unknown origin) assessed as reduction in ATPase activity by biomol green reagent based assayMore data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of p97 (unknown origin) in presence of ATP by Biomol Green Reagent based assayMore data for this Ligand-Target Pair
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
University of Pittsburgh Chemical Diversity Center
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Covalent inhibition of p97 (unknown origin) ATPase activity incubated for 60 mins in presence of ATP by Biomol Green Reagent based microplate reader ...More data for this Ligand-Target Pair











































