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Found 665 for UniProtKB: P56481
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50062005((S)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataKi:  0.148nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50016425((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataKi:  0.191nMAssay Description:Binding affinity measured by inhibiting [3H]Boc[Nle28,31]CCK27-33 specific binding to Cholecystokinin receptor in mouse brain membranes at a KD conce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50281737((R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataKi:  0.200nMAssay Description:The compound was evaluated for the inhibition of binding of [3H]-PD 140376 to Cholecystokinin type B receptor in mouse cortex.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.300nMAssay Description:Potency in displacing [3H]propionyl-Cholecystokinin from mouse brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.491nMAssay Description:Binding affinity measured by inhibiting [3H]Boc[Nle28,31]CCK27-33 specific binding to Cholecystokinin receptor in mouse brain membranes at a KD conce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50230677(CHEMBL3351022)
Affinity DataKi:  0.513nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50285623((R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataKi:  0.520nMAssay Description:Binding affinity towards CCK-B receptor in mouse cerebral cortex membrane using [125I]bolton assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50230683(CHEMBL3351024)
Affinity DataKi:  0.708nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50471066(CHEMBL415936)
Affinity DataKi:  0.741nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50285625((R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataKi:  0.880nMAssay Description:Binding affinity towards CCK-B receptor in mouse cerebral cortex membrane using [125I]bolton assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50213845(CHEMBL14557)
Affinity DataKi:  1nMAssay Description:Inhibition of 20 pM [125I]BH-CCK-8S binding to mouse cortical membrane Cholecystokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50213845(CHEMBL14557)
Affinity DataKi:  1.10nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50230676(CHEMBL3351013)
Affinity DataKi:  1.10nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50213845(CHEMBL14557)
Affinity DataKi:  1.10nMAssay Description:Displacement of binding of [125I]CCK-8S to Cholecystokinin type B receptor in mouse cerebral cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50471067(CHEMBL298521)
Affinity DataKi:  1.20nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50471075(CHEMBL299540)
Affinity DataKi:  1.20nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50230678(CHEMBL287735)
Affinity DataKi:  1.40nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50471065(CHEMBL296167)
Affinity DataKi:  1.60nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50470629(CHEMBL342616)
Affinity DataKi:  1.60nMAssay Description:Inhibition of 20 pM [125I]BH-CCK-8S binding to mouse cortical membrane Cholecystokinin 2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50002477((S)-3-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]pentagastrin from Cholecystokinin receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50230680(CHEMBL3350364)
Affinity DataKi:  2nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226755(CHEMBL415630)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]pentagastrin from Cholecystokinin receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50061220(1-((S)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50230681(CHEMBL3351023)
Affinity DataKi:  2.20nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50470612(CHEMBL436209)
Affinity DataKi:  2.20nMAssay Description:Competition with 20 pM [125I]BH-CCK-8S for Cholecystokinin type B receptor binding sites in mouse cortical homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50470623(CHEMBL140179)
Affinity DataKi:  2.30nMAssay Description:Competition with 20 pM [125I]BH-CCK-8S for Cholecystokinin type B receptor binding sites in mouse cortical homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50470617(CHEMBL137180)
Affinity DataKi:  2.70nMAssay Description:Competition with 20 pM [125I]BH-CCK-8S for Cholecystokinin type B receptor binding sites in mouse cortical homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50024317(3-{2-[2-Amino-3-(1H-indol-3-yl)-propionylamino]-4-...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]pentagastrin from Cholecystokinin receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50470636(CHEMBL343367)
Affinity DataKi:  3.20nMAssay Description:Competition with 20 pM [125I]BH-CCK-8S for Cholecystokinin type B receptor binding sites in mouse cortical homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM81962(S-L-365,260)
Affinity DataKi:  3.70nMAssay Description:Tested for its receptor affinity from competition with 20 pM [125I]BH-CCK-8S for Cholecystokinin type B receptor binding sites in mouse cortical homo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50230689(CHEMBL3351018)
Affinity DataKi:  3.70nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50230687(CHEMBL3351021)
Affinity DataKi:  3.90nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50471076(CHEMBL299387)
Affinity DataKi:  3.90nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM81962(S-L-365,260)
Affinity DataKi:  4nMAssay Description:Displacement of binding of [125I]CCK-8S to Cholecystokinin type B receptor in mouse cerebral cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50470639(CHEMBL433656)
Affinity DataKi:  4nMAssay Description:Competition with 20 pM [125I]BH-CCK-8S for Cholecystokinin type B receptor binding sites in mouse cortical homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50230684(CHEMBL353157 | PD-135118)
Affinity DataKi:  4nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50471072(CHEMBL53237)
Affinity DataKi:  4.10nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50470624(CHEMBL337673)
Affinity DataKi:  4.40nMAssay Description:Competition with 20 pM [125I]BH-CCK-8S for Cholecystokinin type B receptor binding sites in mouse cortical homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50471068(CHEMBL298551)
Affinity DataKi:  4.5nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50421390(CHEMBL24313)
Affinity DataKi:  5nMAssay Description:Inhibition of 20 pM [125I]BH-CCK-8S binding to mouse cortical membrane Cholecystokinin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50421390(CHEMBL24313)
Affinity DataKi:  5.20nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50471071(CHEMBL297480)
Affinity DataKi:  5.40nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50061988(CHEMBL138657 | [(R)-1-((S)-1-Hydroxymethyl-2-pheny...)
Affinity DataKi:  6nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50471073(CHEMBL301777)
Affinity DataKi:  7.60nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50470625(CHEMBL335587)
Affinity DataKi:  7.60nMAssay Description:Competition with 20 pM [125I]BH-CCK-8S for Cholecystokinin type B receptor binding sites in mouse cortical homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50470629(CHEMBL342616)
Affinity DataKi:  7.90nMAssay Description:Competition with 20 pM [125I]BH-CCK-8S for Cholecystokinin type B receptor binding sites in mouse cortical homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50470629(CHEMBL342616)
Affinity DataKi:  7.94nMAssay Description:Competition with 20 pM [125I]BH-CCK-8S for Cholecystokinin type B receptor binding sites in mouse cortical homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50061990((R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataKi:  8.90nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50470634(CHEMBL135350)
Affinity DataKi:  10nMAssay Description:Competition with 20 pM [125I]BH-CCK-8S for Cholecystokinin type B receptor binding sites in mouse cortical homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Parke-Davis Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50470642(CHEMBL421921)
Affinity DataKi:  12nMAssay Description:Competition with 20 pM [125I]BH-CCK-8S for Cholecystokinin type B receptor binding sites in mouse cortical homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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