Compile Data Set for Download or QSAR
Report error Found 148 of affinity data for UniProtKB/TrEMBL: P70597
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252472BDBM50252472(CHEMBL4085914)
Affinity DataIC50: 1.10nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260732BDBM50260732(CHEMBL4105205)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at rat His-tagged EP1 receptor expressed in African green monkey COS1 cells assessed as reduction in PGE2-induced increase in int...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252483BDBM50252483(CHEMBL4081524)
Affinity DataIC50: 6.20nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252452BDBM50252452(CHEMBL4074797)
Affinity DataIC50: 6.40nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260740BDBM50260740(CHEMBL4100262)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at rat His-tagged EP1 receptor expressed in African green monkey COS1 cells assessed as reduction in PGE2-induced increase in int...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240170BDBM50240170(CHEMBL4064816)
Affinity DataIC50: 9.40nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240170BDBM50240170(CHEMBL4064816)
Affinity DataIC50: 9.40nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252462BDBM50252462(CHEMBL4104333)
Affinity DataIC50: 9.90nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260656BDBM50260656(CHEMBL4083796)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at rat His-tagged EP1 receptor expressed in African green monkey COS1 cells assessed as reduction in PGE2-induced increase in int...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119458BDBM119458(US8680120, 9-32)
Affinity DataIC50: 11nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Fluo-4 NW Calcium Assay Kit ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50160913BDBM50160913(6-[3-(2-Benzyloxy-5-chloro-phenyl)-thiophen-2-yl]-...)
Affinity DataKi:  12nMAssay Description:Binding affinity towards Prostaglandin E receptor was determined in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50259548BDBM50259548(6-(5'-chloro-2'-isobutoxy-biphenyl-2-yl)-pyridine-...)
Affinity DataIC50: 12.6nMAssay Description:Binding affinity to rat EP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252484BDBM50252484(CHEMBL4059569)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119456BDBM119456(US8680120, 9-21)
Affinity DataIC50: 13nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Fluo-4 NW Calcium Assay Kit ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119460BDBM119460(US8680120, 9-43)
Affinity DataIC50: 13nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Fluo-4 NW Calcium Assay Kit ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260658BDBM50260658(CHEMBL4091580)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at rat His-tagged EP1 receptor expressed in African green monkey COS1 cells assessed as reduction in PGE2-induced increase in int...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119471BDBM119471(US8680120, 25-26)
Affinity DataIC50: 17nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119468BDBM119468(US8680120, 25-18)
Affinity DataIC50: 17nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252509BDBM50252509(CHEMBL4060696)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260657BDBM50260657(CHEMBL4062060)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at rat His-tagged EP1 receptor expressed in African green monkey COS1 cells assessed as reduction in PGE2-induced increase in int...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119461BDBM119461(US8680120, 9-44)
Affinity DataIC50: 19nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Fluo-4 NW Calcium Assay Kit ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119453BDBM119453(US8680120, 9-1)
Affinity DataIC50: 21nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Fluo-4 NW Calcium Assay Kit ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260660BDBM50260660(CHEMBL4088835)
Affinity DataIC50: 21nMAssay Description:Antagonist activity at rat His-tagged EP1 receptor expressed in African green monkey COS1 cells assessed as reduction in PGE2-induced increase in int...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119455BDBM119455(US8680120, 9-15)
Affinity DataIC50: 22nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Fluo-4 NW Calcium Assay Kit ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252464BDBM50252464(CHEMBL4081022)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419410BDBM50419410(CHEMBL1915252)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as decrease in prostaglandin E2-induced increase in int...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119479BDBM119479(US8680120, 25-38)
Affinity DataIC50: 22nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119459BDBM119459(US8680120, 9-35)
Affinity DataIC50: 23nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Fluo-4 NW Calcium Assay Kit ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119481BDBM119481(US8680120, 25-41)
Affinity DataIC50: 25nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119473BDBM119473(US8680120, 25-29)
Affinity DataIC50: 26nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119478BDBM119478(US8680120, 25-37)
Affinity DataIC50: 27nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119472BDBM119472(US8680120, 25-28)
Affinity DataIC50: 28nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119482BDBM119482(US8680120, 25-42)
Affinity DataIC50: 28nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260702BDBM50260702(CHEMBL4089536)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at rat His-tagged EP1 receptor expressed in African green monkey COS1 cells assessed as reduction in PGE2-induced increase in int...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252481BDBM50252481(CHEMBL4079088)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252510BDBM50252510(CHEMBL4076413)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252494BDBM50252494(CHEMBL4105272)
Affinity DataIC50: 31nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119470BDBM119470(US8680120, 25-23)
Affinity DataIC50: 32nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252465BDBM50252465(CHEMBL4088913)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119467BDBM119467(US8680120, 25-17)
Affinity DataIC50: 32nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119474BDBM119474(US8680120, 25-31)
Affinity DataIC50: 33nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252492BDBM50252492(CHEMBL4062313)
Affinity DataIC50: 33nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119463BDBM119463(US8680120, 25-11)
Affinity DataIC50: 34nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119457BDBM119457(US8680120, 9-25)
Affinity DataIC50: 35nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Fluo-4 NW Calcium Assay Kit ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119477BDBM119477(US8680120, 25-36)
Affinity DataIC50: 35nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119469BDBM119469(US8680120, 25-19)
Affinity DataIC50: 36nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252508BDBM50252508(CHEMBL4096603)
Affinity DataIC50: 37nMAssay Description:Antagonist activity at rat EP1 receptor expressed in African green monkey COS1 cells assessed as inhibition of prostaglandin-E2-induced increase in i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2019
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119480BDBM119480(US8680120, 25-39)
Affinity DataIC50: 37nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119465BDBM119465(US8680120, 25-13)
Affinity DataIC50: 38nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

TargetProstaglandin E2 receptor EP1 subtype(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119466BDBM119466(US8680120, 25-16)
Affinity DataIC50: 39nMAssay Description:The rat EP1 receptor-expressing cells were washed with the assay buffer. 100 μL of a fluorescent calcium indicator (Calcium kit II, Fluo 4 (Doji...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2014
Entry Details
US Patent

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