TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 3.24nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 27.5nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 27.5nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 135nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 145nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 178nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 191nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 282nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 372nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 447nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 646nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 692nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.45E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.55E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 2.14E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 2.45E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 2.51E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 2.63E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 3.02E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 3.09E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 3.09E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 3.31E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 3.47E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 4.07E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 5.25E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 5.89E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 5.89E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 6.92E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 7.76E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 8.13E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 8.71E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 9.33E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Maxi-K (unknown origin) expressed in HEK293 cells measured by thallium flux assayMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Maxi-K (unknown origin) expressed in HEK293 cells measured by thallium flux assayMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.12E+4nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.12E+4nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.17E+4nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.17E+4nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.17E+4nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.23E+4nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.26E+4nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.35E+4nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.35E+4nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.38E+4nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.51E+4nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.51E+4nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.58E+4nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair