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Found 2668 for UniProtKB: Q14164
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  0.199nMAssay Description:Inhibition of human IKKepsilon using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM276896(US10072001, Example 82 | US10259811, Example 82)
Affinity DataIC50:  0.290nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM276896(US10072001, Example 82 | US10259811, Example 82)
Affinity DataIC50:  0.290nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  0.439nMAssay Description:Inhibition of human IKKepsilon using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM276969(US10072001, Example 145 | US10259811, Example 145)
Affinity DataIC50:  0.481nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM276969(US10072001, Example 145 | US10259811, Example 145)
Affinity DataIC50:  0.481nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM276965(US10072001, Example 141 | US10259811, Example 141)
Affinity DataIC50:  0.687nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM276965(US10072001, Example 141 | US10259811, Example 141)
Affinity DataIC50:  0.687nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM276877(US10072001, Example 63 | US10259811, Example 63)
Affinity DataIC50:  0.710nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM276877(US10072001, Example 63 | US10259811, Example 63)
Affinity DataIC50:  0.710nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM276879(US10072001, Example 65 | US10259811, Example 65)
Affinity DataIC50:  0.770nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM276879(US10072001, Example 65 | US10259811, Example 65)
Affinity DataIC50:  0.770nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM276868(US10072001, Example 54 | US10259811, Example 54)
Affinity DataIC50:  0.810nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM276868(US10072001, Example 54 | US10259811, Example 54)
Affinity DataIC50:  0.810nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM277059(US10072001, Example 251 | US10259811, Example 251)
Affinity DataIC50:  0.815nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM277059(US10072001, Example 251 | US10259811, Example 251)
Affinity DataIC50:  0.815nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM277037(US10072001, Example 229 | US10259811, Example 229)
Affinity DataIC50:  0.851nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM277037(US10072001, Example 229 | US10259811, Example 229)
Affinity DataIC50:  0.851nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM277778(5-(4-((3-methoxy-4-(4-methylpiperazin-1-yl)phenyl)...)
Affinity DataIC50:  1nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM277790(5-(4-((4-(4-methylpiperazin-1-yl)phenyl)amino)-1,3...)
Affinity DataIC50:  1nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM277796(5-(4-((4-(piperazin-1-yl)phenyl)amino)-1,3,5-triaz...)
Affinity DataIC50:  1nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM277944((S)-2-((3,3-difluoro-1-(4H-1,2,4-triazole-3-carbon...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278007(2-(((3R,4S)-3-fluoro-1-(2-hydroxyacetyl)piperidin-...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278038(2-(((S)-3,3-difluoro-1-(4H-1,2,4-triazole-3-carbon...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278039(2-(((S)-3,3-difluoro-1-(2-hydroxyacetyl)piperidin-...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278079((S)-2-((1-acetyl-3,3-difluoropiperidin-4-yl)oxy)-5...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278080((S)-2-((1-acetyl-3,3-difluoropiperidin-4-yl)oxy)-5...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278081((S)-2-((3,3-difluoro-1-formylpiperidin-4-yl)oxy)-5...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278082((S)-2-((3,3-difluoro-1-formylpiperidin-4-yl)oxy)-5...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278083(2-(((3R,4S)-3-fluoro-1-(2-hydroxyacetyl)piperidin-...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278084(2-(((3R,4S)-3-fluoro-1-(2-hydroxyacetyl)piperidin-...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278103(2-(((3R,4S)-3-fluoro-1-(2-hydroxyacetyl)piperidin-...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278268(2-(((3R,4S)-3-fluoro-1-(5-methyl-4H-1,2,4-triazole...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278275(2-(((3R,4S)-3-fluoro-1-((S)-2-hydroxypropanoyl)pip...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278276(2-(((3R,4S)-3-fluoro-1-((S)-2-hydroxypropanoyl)pip...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278278(5-(4-((4-((S)-2,4-dimethylpiperazin-1-yl)phenyl)am...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278279(5-(4-((4-((S)-2,4-dimethylpiperazin-1-yl)phenyl)am...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278286(5-(4-((4-((S)-2,4-dimethylpiperazin-1-yl)-3-methox...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278293(2-(((3R,4S)-1-((S)-2,3-dihydroxypropanoyl)-3-fluor...)
Affinity DataIC50: <1nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM144137(US8969335, A74)
Affinity DataIC50:  1nMpH: 7.5 T: 2°CAssay Description:1 nM IKKe, 800 nM biotinylated IkBalpha(19-42) peptide (Biotin-C6-C6-GLKKERLLDDRHDSGLDSMKDEE) and 10 μM ATP (spiked with 0.3 uCi of 33P-ATP/well) ar...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278167(2-(((3R,4S)-3-fluoro-1-((S)-2-hydroxypropanoyl)pip...)
Affinity DataIC50:  1nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278170(2-(((3R,4S)-3-fluoro-1-(2-hydroxyacetyl)piperidin-...)
Affinity DataIC50:  1nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278171(5-(4-((3-(difluoromethoxy)-4-(4-(oxetan-3-yl)piper...)
Affinity DataIC50:  1nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278172(2-(((3R,4S)-3-fluoro-1-(2-hydroxyacetyl)piperidin-...)
Affinity DataIC50:  1nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278173(5-(4-((3-(difluoromethoxy)-4-(4-(oxetan-3-yl)piper...)
Affinity DataIC50:  1nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278174(2-(((3R,4S)-3-fluoro-1-((S)-2-hydroxypropanoyl)pip...)
Affinity DataIC50:  1nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278176(2-(((3R,4S)-1-((S)-2,3-dihydroxypropanoyl)-3-fluor...)
Affinity DataIC50:  1nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278178(2-(((3R,4S)-3-fluoro-1-((S)-2-hydroxypropanoyl)pip...)
Affinity DataIC50:  1nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278187(2-(((3R,4S)-1-((S)-2,3-dihydroxypropanoyl)-3-fluor...)
Affinity DataIC50:  1nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM278074(2-(((3R,4S)-3-fluoro-1-formylpiperidin-4-yl)oxy)-5...)
Affinity DataIC50:  1nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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