Compile Data Set for Download or QSAR
maximum 50k data
Found 126 of affinity data for UniProtKB/TrEMBL: Q2NLC1
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM25400((2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-y...)
Affinity DataKi:  808nMAssay Description:Displacement of [3H]2-[p-(2-carboxyethyl)phenylethylamino]-5-N-ethylcarboxamidoadenosine from mouse A2A adenosine receptor expressed in HEK293 cell m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50397728(CHEMBL2181976)
Affinity DataKi:  830nMAssay Description:Displacement of [3H] ZM241385 from mouse adenosine A2A receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50085658((2R,3R,4S,5R)-2-(2-Chloro-6-cyclopentylamino-purin...)
Affinity DataKi:  988nMAssay Description:Displacement of [3H]2-[p-(2-carboxyethyl)phenylethylamino]-5-N-ethylcarboxamidoadenosine from mouse A2A adenosine receptor expressed in HEK293 cell m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50118812((2S,3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-iodo-benzylami...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5'-N-ethylcarboxamidoadenosine from mouse recombinant adenosine A2A receptor expressed in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50163031((1S,2R,3S,4R,5S)-4-(2-chloro-6-(2,2-diphenylethyla...)
Affinity DataKi:  1.81E+3nMAssay Description:Displacement of [3H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5'-N-ethylcarboxamidoadenosine from mouse recombinant adenosine A2A receptor expressed in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50517307(CHEMBL4463802)
Affinity DataKi:  2.65E+3nMAssay Description:Displacement of [3H]2-[p-(2-carboxyethyl)phenylethylamino]-5-N-ethylcarboxamidoadenosine from mouse A2A adenosine receptor expressed in HEK293 cell m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50517302(CHEMBL4562258)
Affinity DataKi:  3.99E+3nMAssay Description:Displacement of [3H]2-[p-(2-carboxyethyl)phenylethylamino]-5-N-ethylcarboxamidoadenosine from mouse A2A adenosine receptor expressed in HEK293 cell m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50100418((1S,2R,3S,4R,5S)-4-(6-(3-iodobenzylamino)-2-chloro...)
Affinity DataKi:  5.35E+3nMAssay Description:Displacement of [3H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5'-N-ethylcarboxamidoadenosine from mouse recombinant adenosine A2A receptor expressed in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50163025((1S,2R,3S,4R,5S)-4-(6-(3-bromobenzylamino)-2-chlor...)
Affinity DataKi:  6.39E+3nMAssay Description:Displacement of [3H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5'-N-ethylcarboxamidoadenosine from mouse recombinant adenosine A2A receptor expressed in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM21221((2S,3S,4R,5R)-5-(2-chloro-6-{[(3-iodophenyl)methyl...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5'-N-ethylcarboxamidoadenosine from mouse recombinant adenosine A2A receptor expressed in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50086170((4-Cyano-phenyl)-carbamic acid 4-(2,6-dioxo-1,3-di...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]MSX-2 from recombinant mouse A2A adenosine receptor expressed in CHO cell membranes measured after 60 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50042209(4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]MSX-2 from recombinant mouse A2A adenosine receptor expressed in CHO cell membranes measured after 60 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50163020((1S,2R,3S,4R,5S)-4-(6-(3-chlorobenzylamino)-2-chlo...)
Affinity DataKi:  1.04E+4nMAssay Description:Displacement of [3H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5'-N-ethylcarboxamidoadenosine from mouse recombinant adenosine A2A receptor expressed in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50100416((1S,2R,3S,4R,5S)-4-(2-Chloro-6-methylamino-purin-9...)
Affinity DataKi:  2.04E+4nMAssay Description:Displacement of [3H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5'-N-ethylcarboxamidoadenosine from mouse recombinant adenosine A2A receptor expressed in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50163004((1S,2R,3S,4R,5S)-4-(2-chloro-6-(2-phenylcyclopropy...)
Affinity DataKi:  3.82E+4nMAssay Description:Displacement of [3H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5'-N-ethylcarboxamidoadenosine from mouse recombinant adenosine A2A receptor expressed in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM50163014((1S,2R,3S,4R,5S)-4-(6-(2,5-dimethoxybenzylamino)-2...)
Affinity DataKi:  4.47E+4nMAssay Description:Displacement of [3H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5'-N-ethylcarboxamidoadenosine from mouse recombinant adenosine A2A receptor expressed in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474329(7-(3-fluoro-1H-pyrazol-1-yl)-2-((3-fluoropyridin- ...)
Affinity DataIC50:  0.200nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474284(7-(4-fluorophenyl)-2-((3-fluoropyridin-2-yl) methy...)
Affinity DataIC50:  0.300nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474223(2-(2,6-difluorobenzyl)-8-(2-(dimethylamino) pyridi...)
Affinity DataIC50:  0.400nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474328(7-(4-fluorophenyl)-2-(2-methoxyethyl)-8-(3-met hyl...)
Affinity DataIC50:  0.400nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474287(2-((3-(difluoromethoxy)pyridin-2-yl)methyl)-7- (4-...)
Affinity DataIC50:  0.400nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474330(7-(4-fluoro-1H-pyrazol-1-yl)-2-((3-fluoropyridin- ...)
Affinity DataIC50:  0.5nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474281(7-(4-fluorophenyl)-2-((3-fluoropyridin-2-yl) methy...)
Affinity DataIC50:  0.600nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474233(5-[5-amino-7-(4-fluorophenyl)-2-[(3-fluoropyrid in...)
Affinity DataIC50:  0.800nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474222(5-(5-amino-2-(2,6-difluorobenzyl)-7-(4- fluorophen...)
Affinity DataIC50:  0.800nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474309(2-((3-fluoropyridin-2-yl)methyl)-8-(3-methylimi da...)
Affinity DataIC50:  0.800nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474292(5-(5-am i no-2-(2,6-difluorobenzy1)-7-(oxazol-2- y...)
Affinity DataIC50:  0.900nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474315(7-(4-fluorophenyl)-8-(3-methylimidazo[1,2-a] pyrid...)
Affinity DataIC50:  1nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474316(7-(4-fluorophenyl)-8-(3-methylimidazo[l,2-a] pyrid...)
Affinity DataIC50:  1nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474288(2-((3-(difluoromethoxy)pyridin-2-yl)methyI)-8- (im...)
Affinity DataIC50:  1.20nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474300(7-(4-fluorophenyl)-2-((3-fluoropyridin-2-yl) methy...)
Affinity DataIC50:  1.30nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474245(2-(2,6-difluorobenzyl)-7-(4-fluorophenyl)-8-(2- me...)
Affinity DataIC50:  1.5nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474335((S)-7-(4-fluorophenyl)-8-(3-methylimidazo[1,2-a] p...)
Affinity DataIC50:  2.60nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474299(8-(benzo[d]thiazol-6-yl)-7-(4-fluorophenyl)-2- ((3...)
Affinity DataIC50:  2.60nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474334(2-(2,6-difluorobenzyl)-8-(3-methylimidazo[l,2-a] p...)
Affinity DataIC50:  2.90nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474258(5-[5-amino-7-(4-fluorophenyl)-2-[(3-fluoropyrid in...)
Affinity DataIC50:  2.90nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474230(5-(5-amino-7-(4-fluorophenyl)-2-((3-fluoropyrid in...)
Affinity DataIC50:  3.40nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474310(2-((3*fluoropyridin-2-yl)methyl)-N7,N7-dimethy l-8...)
Affinity DataIC50:  3.5nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474301(2-((3-fluoropyridin-2-yl)methyl)-8-(1-methyl-1H- b...)
Affinity DataIC50:  3.5nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474337(7-(azetidin-l-yl)-2-(2,6-difluorobenzyl)-8-(3-met ...)
Affinity DataIC50:  3.90nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474293(5-(5-amino-2-((3-fluoropyridin-2-yl)methyl)-7- (ox...)
Affinity DataIC50:  4.90nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474224(5-(5-amino-2-[[3-(difluoromethoxy)pyridin-2-yl] me...)
Affinity DataIC50:  4.90nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474302(2-(2,6-difluorobenzyl)-8-(1-methyl-1H-benzo[d] imi...)
Affinity DataIC50:  5.10nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474263(5-(5-amino-7-(4-fluorophenyl)-2-((3-fluoropyrid in...)
Affinity DataIC50:  5.10nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474229(7-(4-fluorophenyl)-2-((3-fluoropyridin-2-yl) methy...)
Affinity DataIC50:  5.40nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474314((R)-7-(4-fluorophenyl)-8-(1-methyl-1H-benzo[d] imi...)
Affinity DataIC50:  5.70nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474273(5-(5-amino-2-(2,6-difluorobenzyl)-7-(thiazol-2- yl...)
Affinity DataIC50:  5.90nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474285(5-(5-amino-2-[[3-(difluoromethoxy)pyridin-2-yl] me...)
Affinity DataIC50:  6.40nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474231(6-[[5-amino-7-(4-fluorophenyl)-8-[imidazo[1,2-a] p...)
Affinity DataIC50:  7.30nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Mus musculus)
Medical College Of Wisconsin

Curated by ChEMBL
LigandPNGBDBM474305(5-(5-amino-7-(4-fluorophenyl)-2-((3-fluoropyrid in...)
Affinity DataIC50:  8.90nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
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