TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 0.230nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse BMDM cells assessed as reduction in ATP induced IL-1beta release pretreated for 15 mi...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 0.390nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse BMDM cells assessed as reduction in ATP induced IL-1beta release pretreated for 15 mi...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta level incubated for 1 hr followed by ...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774A.1 cells assessed as reduction in IL-1beta level preincubated for 30 mins follow...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 in LPS/ATP-treated mouse bone marrow derived macrophages assessed as reduction in NLRP3 inflammasome activation by measuring redu...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 in mouse BMDM cells preincubated for 30 mins followed by ATP addition by ELISA analysisMore data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-stimulated mouse BMDM assessed as reduction in NLRP3 inflammasome-induced IL-1beta production prei...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated mouse BMDM cells assessed as inhibition of LPS and nigericin-induced IL-1beta pr...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 in mouse BMDMsMore data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse bone marrow derived macrophages assessed as reduction in IL-1beta level preincubated ...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of NLRP3 inflammasome in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 30 mins followed by A...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated mouse J774A.1 cells assessed as decrease in IL-1beta level pretreated for 0.5 hr...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/nigericin-treated mouse J774A.1 cells assessed as decrease in LDH release pretreated for 0.5 hrs f...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of NLRP3 in mouse peritoneal macrophages assessed as inhibition of LPS and ATP-induced IL-1beta production pre-stimulated with LPS for 4.5...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of NLRP3 in mouse peritoneal macrophages assessed as inhibition of LPS and ATP-induced IL-1beta production pre-stimulated with LPS for 4.5...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse bone marrow derived macrophages assessed as reduction in IL-1beta level preincubated ...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of NLRP3 induced IL-1beta release in LPS/nigericin-treated mouse BMDM cells preincubated with LPS for 3 hrs followed by compound addition ...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 74nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of NLRP3 in mouse J774A.1 cells infected with FLA-ST assessed as inhibition of LPS- induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS and ATP-stimulated mouse whole blood assessed as reduction in IL-1beta release preincubated for 3 ...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of NLRP3 in mouse BMDM assessed as reduction in LPS-stimulated IL-1beta levels pre-incubated with LPS for 4.5 hrs followed by incubation f...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of NLRP3 inflammasome in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 30 mins followed by A...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of NLRP3 inflammasome in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 30 mins followed by A...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 141nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 151nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of NLRP3 inflammasome in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 30 mins followed by A...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of NLRP3 inflammasome in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 30 mins followed by A...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 195nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of NLRP3 inflammasome in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 30 mins followed by A...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of NLRP3 inflammasome in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 30 mins followed by A...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 234nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 1 hr follo...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of NLRP3 inflammasome in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 30 mins followed by A...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of NLRP3 inflammasome in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 30 mins followed by A...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of NLRP3 inflammasome in LPS-primed mouse J774.A1 cells assessed as reduction in IL-1beta secretion preincubated for 30 mins followed by A...More data for this Ligand-Target Pair
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
Hospital Universitario Santa Cristina
Curated by ChEMBL
Hospital Universitario Santa Cristina
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of NLRP3 in mouse J774A.1 cells assessed as inhibition of LPS and ATP-induced IL-1beta production pre-stimulated with LPS for 4.5 hrs befo...More data for this Ligand-Target Pair