Compile Data Set for Download or QSAR
maximum 50k data
Found 127 of affinity data for UniProtKB/TrEMBL: Q8WU89
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009575(CHEMBL3234446)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009560(CHEMBL3234454)
Affinity DataKi:  89nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009571(CHEMBL3234461)
Affinity DataKi:  180nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009572(CHEMBL3234462)
Affinity DataKi:  270nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009558(CHEMBL3234452)
Affinity DataKi:  310nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009559(CHEMBL3234453)
Affinity DataKi:  400nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009580(CHEMBL3234445)
Affinity DataKi:  430nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009567(CHEMBL3234458)
Affinity DataKi:  450nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009576(CHEMBL3234447)
Affinity DataKi:  690nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009574(CHEMBL3234464)
Affinity DataKi:  850nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009573(CHEMBL3234463)
Affinity DataKi:  960nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009566(CHEMBL3234457)
Affinity DataKi:  970nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009570(CHEMBL3234460)
Affinity DataKi:  980nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009569(CHEMBL3234459)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009579(CHEMBL3234448)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009577(CHEMBL3234450)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009578(CHEMBL3234449)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009557(CHEMBL3234451)
Affinity DataKi:  9.00E+3nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009564(CHEMBL3234456)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009563(CHEMBL3234455)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610888(4-(2,6-Dimethoxyphenyl)-5-(5-methylfuran-2-yl)-4H-...)
Affinity DataEC50:  31nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610889(2-({[4-(2,6-Dimethoxyphenyl)-5-(5-methylfuran-2-yl...)
Affinity DataEC50:  1nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610890(7-Chloro-2-({[4-(2,6-dimethoxyphenyl)-5-(5-methylf...)
Affinity DataEC50:  2nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610891(Ethyl {[4-(2,6-dimethoxyphenyl)-5-(5-methylfuran-2...)
Affinity DataEC50:  122nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610892(US10626096, Example 5 | {[4-(2,6-Dimethoxyphenyl)-...)
Affinity DataEC50:  26nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610893(4-(2,6-Dimethoxyphenyl)-3-(5-methylfuran-2-yl)-4H-...)
Affinity DataEC50:  703nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610894(US10626096, Example 7 | [4-(2,6-Dimethoxyphenyl)-5...)
Affinity DataEC50:  815nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610895(US10626096, Example 8)
Affinity DataEC50:  1.57E+3nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610896((2E)-3-[4-(2,6-Dimethoxyphenyl)-5-(5-methylfuran-2...)
Affinity DataEC50:  18nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610897(US10626096, Example 10)
Affinity DataEC50:  192nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610898(US10626096, Example 11 | [2-({[4-(2,6-Dimethoxyphe...)
Affinity DataEC50:  5nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610899(Ethyl 3-[4-(2,6-dimethoxyphenyl)-5-(5-methylfuran-...)
Affinity DataEC50:  701nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610900(3-[4-(2,6-Dimethoxyphenyl)-5-(5-methylfuran-2-yl)-...)
Affinity DataEC50:  159nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610901(6-({[4-(2,6-Dimethoxyphenyl)-5-(5-methylfuran-2-yl...)
Affinity DataEC50:  424nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610902(6-({[4-(2,6-Dimethoxyphenyl)-5-(5-methylfuran-2-yl...)
Affinity DataEC50:  164nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610903(5-({[4-(2,6-Dimethoxyphenyl)-5-(5-methylfuran-2-yl...)
Affinity DataEC50:  314nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610904(US10626096, Example 17)
Affinity DataEC50:  1.41E+3nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610905(4-({[4-(2,6-Dimethoxyphenyl)-5-(5-methylfuran-2-yl...)
Affinity DataEC50:  561nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610906((2E)-3-[4-(2,6-Dimethoxyphenyl)-5-(5-methylfuran-2...)
Affinity DataEC50:  171nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610907((3E)-4-[4-(2,6-Dimethoxyphenyl)-5-(5-methylfuran-2...)
Affinity DataEC50:  729nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610908((2E)-3-[4-(2,6-Dimethoxyphenyl)-5-(5-methylfuran-2...)
Affinity DataEC50:  539nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610909(US10626096, Example 22)
Affinity DataEC50:  87nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610910((3E)-4-[4-(2,6-Dimethoxyphenyl)-5-(5-methylfuran-2...)
Affinity DataEC50:  271nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610911(4-[4-(2,6-Dimethoxyphenyl)-5-(5-methylfuran-2-yl)-...)
Affinity DataEC50:  751nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610912(4-[4-(2,6-Dimethoxyphenyl)-5-(5-methylfuran-2-yl)-...)
Affinity DataEC50:  1.72E+3nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610913(US10626096, Example 26)
Affinity DataEC50:  57nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610914(US10626096, Example 27)
Affinity DataEC50:  2.87E+3nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610915(US10626096, Example 28)
Affinity DataEC50:  1.42E+3nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610916(US10626096, Example 29)
Affinity DataEC50:  812nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM610917(US10626096, Example 30)
Affinity DataEC50:  332nMAssay Description:The apelin receptor agonist activity of the compound represented by formula (I) or (II) of the present invention was measured by cell-based assay for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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