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Found 29 of affinity data for UniProtKB/TrEMBL: Q99P79
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50506039(CHEMBL1324296)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]TCDD from mouse AhR expressed in mouse Hepa1c1c7 cells cytosol incubated for 2 hrs by competitive radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50605060(CHEMBL5198290)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]TCDD from mouse AhR expressed in mouse Hepa1c1c7 cells cytosol incubated for 2 hrs by competitive radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50605061(CHEMBL5179114)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]TCDD from mouse AhR expressed in mouse Hepa1c1c7 cells cytosol incubated for 2 hrs by competitive radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50439845(CHEMBL2420083)
Affinity DataIC50:  21nMAssay Description:Displacement of 2-azido-3-[125I]7,8-dibromodibenzo-pdioxin from C57BL/6J mouse liver AhR incubated for 20 mins by gamma counting based autoradiograph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50014323(2-PHENYL-4H-BENZO[H]CHROMEN-4-ONE | 2-Phenyl-benzo...)
Affinity DataIC50:  25nMAssay Description:Displacement of 2-azido-3-[125I]7,8-dibromodibenzo-pdioxin from C57BL/6J mouse liver AhR incubated for 20 mins by gamma counting based autoradiograph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM92709(Photoaffinity ligand, 6)
Affinity DataKd:  8.10nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM92710(Photoaffinity ligand, 7)
Affinity DataKd:  113nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM92711(Photoaffinity ligand, 8)
Affinity DataKd:  11nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50015301(CHEMBL3263111)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at AHR in FVB/N mouse primary mammary epithelial cells assessed as blockade of mammary branching morphogenesis after 144 hrs by micr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50015302(CHEMBL3263112)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at AHR in FVB/N mouse primary mammary epithelial cells assessed as blockade of mammary branching morphogenesis after 144 hrs by micr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50015303(CHEMBL3263118)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at AHR in FVB/N mouse primary mammary epithelial cells assessed as blockade of mammary branching morphogenesis after 144 hrs by micr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50015304(CHEMBL3263119)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at AHR in FVB/N mouse primary mammary epithelial cells assessed as blockade of mammary branching morphogenesis after 144 hrs by micr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50015305(CHEMBL3263120)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at AHR in FVB/N mouse primary mammary epithelial cells assessed as blockade of mammary branching morphogenesis after 144 hrs by micr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50357322(CHEMBL1916880)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Ah receptor in genetically engineered mouse cells expressing firefly luciferase gene by CALUX transactivational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50357333(CHEMBL1916891)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Ah receptor in genetically engineered mouse cells expressing firefly luciferase gene by CALUX transactivational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50357339(CHEMBL1916897)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Ah receptor in genetically engineered mouse cells expressing firefly luciferase gene by CALUX transactivational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50357344(CHEMBL1916902)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Ah receptor in genetically engineered mouse cells expressing firefly luciferase gene by CALUX transactivational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM23927(2,3,7,8-Tetrachlorodibenzo-p-dioxin | 2,3,7,8-tetr...)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at Ah receptor in genetically engineered mouse cells expressing firefly luciferase gene by CALUX transactivational assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50506039(CHEMBL1324296)
Affinity DataKd:  3nMAssay Description:Displacement of [3H]TCDD from mouse AhRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50239186(1,1-Bis(3''-Indolyl)Methane | 3,3''-Diindolylmetha...)
Affinity DataEC50:  7.80E+4nMAssay Description:Displacement of 2-azido-3-[125I]7,8-dibromodibenzo-pdioxin from C57BL/6J mouse liver AhR relative to TCDDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50239186(1,1-Bis(3''-Indolyl)Methane | 3,3''-Diindolylmetha...)
Affinity DataKd:  90nMAssay Description:Displacement of 2-azido-3-[125I]7,8-dibromodibenzo-pdioxin from C57BL/6J mouse liver AhRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50602335(CHEMBL5186309)
Affinity DataEC50:  0.0580nMAssay Description:Activation of AhR in mouse NIH3T3 cells assessed as induction of XRE-dependent reporter activity incubated for 4 hrs by Renilla/Firefly based dual-lu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50602335(CHEMBL5186309)
Affinity DataEC50:  71nMAssay Description:Activation of AhR in mouse Hepa1c1c7 cells assessed as induction of XRE-dependent reporter activity incubated for 4 hrs by Renilla/Firefly based dual...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM92708(Photoaffinity ligand, 5)
Affinity DataKd:  13nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM92707(Photoaffinity ligand, 4)
Affinity DataKd:  0.760nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM92706(Photoaffinity ligand, 3)
Affinity DataKd:  0.490nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM50506039(CHEMBL1324296)
Affinity DataEC50:  10nMAssay Description:Agonist activity at AhR in mouse Hepa2Dluc cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM92704(Photoaffinity ligand, 1)
Affinity DataKd:  0.440nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Mus musculus (Mouse))
Palack£

Curated by ChEMBL
LigandPNGBDBM92705(Photoaffinity ligand, 2)
Affinity DataKd:  2.10nMpH: 7.5 T: 2°CAssay Description:The equilibrium dissocation constants, KD values for the photoaffinity ligands were determined by a competitive binding assay. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed