Affinity DataKi: 0.00230nMAssay Description:Inhibition of trypsin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Inhibition of human cationic trypsin using Boc-VPR-MCA as substrate measured every 30 secs for 10 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Inhibition of beta-trypsin (unknown origin) using Bz-FVRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.0450nMAssay Description:Compound was tested in vitro for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0450nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0450nMAssay Description:Tested for selectivity against trypsinChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0540nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su...More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Compound was tested for inhibition of Sunflower beta-trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibition of trypsin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Inhibition of trypsin (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Inhibition of beta-trypsin (unknown origin) using Bz-FVRpNA substrate by spectrophotometry methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su...More data for this Ligand-Target Pair
Affinity DataKi: 0.180nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 uL) was mixed with 20 uM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 uL) mixed ...More data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.180nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ...More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su...More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.210nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su...More data for this Ligand-Target Pair
Affinity DataKi: 0.210nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 uL) was mixed with 20 uM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 uL) mixed ...More data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su...More data for this Ligand-Target Pair
Affinity DataKi: 0.210nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL) was mixed with 20 μM fluorescence enzyme substrate (Boc-Phe-Ser-Arg-AMC, 50 ...More data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:The compound was tested for its ability to inhibit thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.240nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su...More data for this Ligand-Target Pair
Affinity DataKi: 0.240nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su...More data for this Ligand-Target Pair
Affinity DataKi: 0.25nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su...More data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:The compound was tested for its ability to inhibit thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Compound was evaluated for its binding affinity to the trypsin enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:In vitro inhibition constant (Ki) against human human trypsin was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.370nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.380nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su...More data for this Ligand-Target Pair
Affinity DataKi: 0.380nMpH: 8.0Assay Description:Using a 96 well plate (#3915, Costar), a test compound (25 μL), 400 mM Tris-HCl buffer (pH 8.0, 25 μL) and 0.5 mg/mL fluorescence enzyme su...More data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition assay using human trysin.More data for this Ligand-Target Pair