TargetGlutamate receptor ionotropic, NMDA 1 [F484A,T518L]/3A(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 3.50E+4nM ΔG°: -25.4kJ/mole IC50: 9.70E+4nMpH: 7.4 T: 2°CAssay Description:Two-electrode voltage clamp (TEVC) recordings were performed on Xenopus oocytes at room temperature 3-6 days postinjection using an OC-725C TEVC ampl...More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2B receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 95nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2B receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2B receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 820nMAssay Description:The compound was tested in vitro for activity against NR1A/2B sub type of NMDA receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Compound was tested in vitro for inhibition of NMDA response at cloned NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2B receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40E+3nMAssay Description:Compound was tested in vitro for inhibition of NMDA response at cloned NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2B receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2B receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+4nMAssay Description:Compound was tested in vitro for inhibition of NMDA response at cloned NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+4nMAssay Description:Compound was tested in vitro for inhibition of NMDA response at cloned NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+4nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2B receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+4nMAssay Description:Compound was tested in vitro for inhibition of NMDA response at cloned NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Compound was tested in vitro for inhibition of NMDA response at cloned NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+4nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2B receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+4nMAssay Description:Compound was tested in vitro for inhibition of NMDA response at cloned NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+4nMAssay Description:Compound was tested in vitro for inhibition of NMDA response at cloned NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+4nMAssay Description:Compound was tested in vitro for inhibition of NMDA response at cloned NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+4nMAssay Description:Compound was tested in vitro for inhibition of NMDA response at cloned NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80E+4nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of NMDA response at NR1A/2B receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Compound was tested in vitro for inhibition of NMDA response at cloned NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of NMDA responses at NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair