Compile Data Set for Download or QSAR
maximum 50k data
Found 80 of affinity data for UniProtKB/TrEMBL: Q9UEW9
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206401(CHEMBL246321 | N-((S)-1-amino-3-(4-hydroxyphenyl)-...)
Affinity DataKi:  0.311nMAssay Description:Displacement of [125I]-hCG from LH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505809(CHEMBL4460075)
Affinity DataIC50:  81nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50383229(CHEMBL2032175)
Affinity DataIC50:  95nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)
Affinity DataIC50:  96nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)
Affinity DataIC50:  97nMAssay Description:Negative allosteric modulation of human luteinizing hormone receptor assessed as reduction in glycoprotein human luteinizing hormone-induced agonist ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505791(CHEMBL4587440)
Affinity DataIC50:  102nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505799(CHEMBL4573509)
Affinity DataIC50:  107nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505796(CHEMBL4531781)
Affinity DataIC50:  127nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505785(CHEMBL4443605)
Affinity DataIC50:  174nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505783(CHEMBL4458424)
Affinity DataIC50:  185nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505811(CHEMBL4461980)
Affinity DataIC50:  193nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)
Affinity DataIC50:  200nMAssay Description:Negative allosteric modulation of human luteinizing hormone receptor assessed as reduction in glycoprotein human luteinizing hormone-induced agonist ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505797(CHEMBL4522381)
Affinity DataIC50:  207nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505798(CHEMBL4581889)
Affinity DataIC50:  275nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505812(CHEMBL4555151)
Affinity DataIC50:  312nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505795(CHEMBL4579421)
Affinity DataIC50:  332nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505793(CHEMBL4593222)
Affinity DataIC50:  378nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505789(CHEMBL4471621)
Affinity DataIC50:  403nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505804(CHEMBL4590976)
Affinity DataIC50:  486nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505813(CHEMBL4580951)
Affinity DataIC50:  580nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)
Affinity DataIC50:  650nMAssay Description:Negative allosteric modulation of human luteinizing hormone receptor assessed as reduction in Org 43553-induced agonist activity preincubated for 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)
Affinity DataIC50:  1.20E+3nMAssay Description:Negative allosteric modulation of human luteinizing hormone receptor assessed as reduction in Org 43553-induced agonist activity preincubated for 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)
Affinity DataIC50:  1.50E+3nMAssay Description:Negative allosteric modulation of human luteinizing hormone receptor assessed as reduction in Org 43553-induced agonist activity preincubated for 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)
Affinity DataIC50:  1.50E+3nMAssay Description:Negative allosteric modulation of human luteinizing hormone receptor assessed as reduction in Org 43553-induced agonist activity preincubated for 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505786(CHEMBL4560733)
Affinity DataIC50:  1.62E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505794(CHEMBL4456365)
Affinity DataIC50:  1.68E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)
Affinity DataIC50:  1.70E+3nMAssay Description:Negative allosteric modulation of human luteinizing hormone receptor assessed as reduction in Org 43553-induced agonist activity preincubated for 20 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505808(CHEMBL4464604)
Affinity DataIC50:  1.85E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)
Affinity DataIC50:  2.20E+3nMAssay Description:Negative allosteric modulation of human luteinizing hormone receptor assessed as reduction in glycoprotein human luteinizing hormone-induced agonist ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)
Affinity DataIC50:  2.20E+3nMAssay Description:Negative allosteric modulation of human luteinizing hormone receptor assessed as reduction in glycoprotein human luteinizing hormone-induced agonist ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50256858(CHEMBL474041 | Cyclopentyl-carbamic acid [1,1',3',...)
Affinity DataIC50:  2.30E+3nMAssay Description:Displacement of [3H]Org43553 from human luteinizing hormone receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505810(CHEMBL4551301)
Affinity DataIC50:  2.31E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)
Affinity DataIC50:  2.50E+3nMAssay Description:Negative allosteric modulation of human luteinizing hormone receptor assessed as reduction in glycoprotein human luteinizing hormone-induced agonist ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505802(CHEMBL4468163)
Affinity DataIC50:  2.61E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505800(CHEMBL4588196)
Affinity DataIC50:  3.13E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505801(CHEMBL4570127)
Affinity DataIC50:  3.24E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505792(CHEMBL4471875)
Affinity DataIC50:  3.32E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505815(CHEMBL4468307)
Affinity DataIC50:  3.65E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505816(CHEMBL4573451)
Affinity DataIC50:  5.18E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505788(CHEMBL4449797)
Affinity DataIC50:  6.79E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505806(CHEMBL4471103)
Affinity DataIC50:  7.47E+3nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505790(CHEMBL4553576)
Affinity DataIC50: >1.60E+4nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505807(CHEMBL4463418)
Affinity DataIC50: >1.65E+4nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505805(CHEMBL4563783)
Affinity DataIC50: >1.65E+4nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505803(CHEMBL4524393)
Affinity DataIC50: >1.65E+4nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505814(CHEMBL4458027)
Affinity DataIC50: >1.65E+4nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50505784(CHEMBL4464888)
Affinity DataIC50: >1.65E+4nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50189779(CHEMBL377399 | N-tert-butyl-5-amino-4-(3-methoxyph...)
Affinity DataEC50:  800nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206403(CHEMBL269261 | N-((S)-1-amino-3-(4-tert-butoxyphen...)
Affinity DataEC50:  1.21E+4nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50206404((S)-N-(1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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