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BindingDB Data by Journal

PMIDDataArticle TitleCitationOrganizationData Download
2795950856Transformation of the Non-Selective Aminocyclohexanol-Based Hsp90 Inhibitor into a Grp94-Seletive Scaffold.BDBACS Chem Biol 12: 244-253 (2017)The University of Kansas2D 3D TSV
2797711524LSD1 Substrate Binding and Gene Expression Are Affected by HDAC1-Mediated Deacetylation.BDBACS Chem Biol 12: 254-264 (2017)Wayne State University2D 3D TSV
2802616241hBfl-1/hNOXA Interaction Studies Provide New Insights on the Role of Bfl-1 in Cancer Cell Resistance and for the Design of Novel Anticancer Agents.BDBACS Chem Biol 12: 444-455 (2017)University of California Riverside2D 3D TSV
2802616722Heat Capacity Changes for Transition-State Analogue Binding and Catalysis with Human 5'-Methylthioadenosine Phosphorylase.BDBACS Chem Biol 12: 464-473 (2017)Albert Einstein College of Medicine2D 3D TSV
280454907An Allosteric Inhibitor Scaffold Targeting the PIF-Pocket of Atypical Protein Kinase C Isoforms.BDBACS Chem Biol 12: 564-573 (2017)Universitätsklinikum Frankfurt2D 3D TSV
280949132Inhibition of Pax2 Transcription Activation with a Small Molecule that Targets the DNA Binding Domain.BDBACS Chem Biol 12: 724-734 (2017)University of Michigan2D 3D TSV
2803298012Ligand Discovery for a Peptide-Binding GPCR by Structure-Based Screening of Fragment- and Lead-Like Chemical Libraries.BDBACS Chem Biol 12: 735-745 (2017)Stockholm University2D 3D TSV
280357962Structural Insights into the Inhibition of Tubulin by the Antitumor Agent 4ß-(1,2,4-triazol-3-ylthio)-4-deoxypodophyllotoxin.BDBACS Chem Biol 12: 746-752 (2017)Huazhong Agricultural University2D 3D TSV
281350689Development of Potent, Selective SRPK1 Inhibitors as Potential Topical Therapeutics for Neovascular Eye Disease.BDBACS Chem Biol 12: 825-832 (2017)Exonate Ltd2D 3D TSV
2819570447Highly Potent Cell-Permeable and Impermeable NanoLuc Luciferase Inhibitors.BDBACS Chem Biol 12: 1028-1037 (2017)Promega Biosciences LLC2D 3D TSV
2832340610Affinity Selection-Mass Spectrometry Identifies a Novel Antibacterial RNA Polymerase Inhibitor.BDBACS Chem Biol 12: 1346-1352 (2017)Merck & Co. Inc2D 3D TSV
283140978Fragment-Sized EthR Inhibitors Exhibit Exceptionally Strong Ethionamide Boosting Effect in Whole-Cell Mycobacterium tuberculosis Assays.BDBACS Chem Biol 12: 1390-1396 (2017)University of Cambridge2D 3D TSV
2828770017Price for Opening the Transient Specificity Pocket in Human Aldose Reductase upon Ligand Binding: Structural, Thermodynamic, Kinetic, and Computational Analysis.BDBACS Chem Biol 12: 1397-1415 (2017)Philipps-Universität Marburg2D 3D TSV
284062894Phylogenomic Analysis of the Microviridin Biosynthetic Pathway Coupled with Targeted Chemo-Enzymatic Synthesis Yields Potent Protease Inhibitors.BDBACS Chem Biol 12: 1538-1546 (2017)University of Helsinki2D 3D TSV
284406167Discovery and Characterization of a Eukaryotic Initiation Factor 4A-3-Selective Inhibitor That Suppresses Nonsense-Mediated mRNA Decay.BDBACS Chem Biol 12: 1760-1768 (2017)BC Cancer Agency2D 3D TSV
284815028Efficient Inhibition of SmNACE by Coordination Complexes Is Abolished by S. mansoni Sequestration of Metal.BDBACS Chem Biol 12: 1787-1795 (2017)University of Strasburg2D 3D TSV
2871918521Small Molecule Enhancement of 20S Proteasome Activity Targets Intrinsically Disordered Proteins.BDBACS Chem Biol 12: 2240-2247 (2017)Michigan State University2D 3D TSV
287964889Direct Interaction of Chivosazole F with Actin Elicits Cell Responses Similar to Latrunculin A but Distinct from Chondramide.BDBACS Chem Biol 12: 2264-2269 (2017)Novartis Pharma AG2D 3D TSV
2879319132Structural Basis of Analog Specificity in PKG I and II.BDBACS Chem Biol 12: 2388-2398 (2017)Baylor College of Medicine2D 3D TSV
2883675431Cell Lysate-Based AlphaLISA Deubiquitinase Assay Platform for Identification of Small Molecule Inhibitors.BDBACS Chem Biol 12: 2399-2407 (2017)University of Delaware2D 3D TSV
288412822Synthetic Lethality Triggered by Combining Olaparib with BRCA2-Rad51 Disruptors.BDBACS Chem Biol 12: 2491-2497 (2017)Istituto Italiano di Tecnologia2D 3D TSV
2884990813Selective Targeting of Bromodomains of the Bromodomain-PHD Fingers Family Impairs Osteoclast Differentiation.BDBACS Chem Biol 12: 2619-2630 (2017)Oxford University2D 3D TSV
2889260520Inhibitors of the Diadenosine Tetraphosphate Phosphorylase Rv2613c of Mycobacterium tuberculosis.BDBACS Chem Biol 12: 2682-2689 (2017)University of Konstanz2D 3D TSV