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Compound Name:

Compounds Sorted by Binding Data per Compound

1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29
30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 78 79 80 81
82 83 84 85 86 87 88 89 90 91 92 93 94 95 96 97 98 99 100 101 102 103 104 105
106 107 108 109 110 111 112 113 114 115 116 117 118 119 120 121 122 123 124
125 127 128 129 130 132 133 134 135 136 137 138 139 140 141 143 144 145 146
147 148 149 150 151 153 154 155 156 159 160 161 163 164 165 168 170 171 173
174 176 178 179 183 184 186 188 189 190 191 192 193 196 198 199 200 203 204
205 206 207 208 209 210 216 220 224 226 227 229 232 237 238 241 243 248 252
253 259 261 270 274 276 277 285 291 303 304 313 318 323 325 328 333 335 337
339 341 353 360 361 365 389 393 398 401 413 433 442 444 445 446 447 448 451
453 454 455 457 458 460 463 465 467 473 477 478 482 484 499 504 505 506 517
521 525 543 549 551 554 591 606 663 691 708 796 804 821 825 833 842 847 854
855 861 873 879 883 887 913 914 925 926 938 947 1010 1027 1050 1052 1081 1082
1099 1115 1130 1133 1206 1262 1543 1639 1903 2029
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Enz. Inhib. Data
ITC Data
Binding Targets
Alternate Compound Names
89 Ki 5 IC50 6 Kd
  • β-Carbonic anhydrase 2 (CA 2)
  • Alpha carbonic anhydrase
  • Astrosclerin-3
  • Beta-carbonic anhydrase
  • Carbonate dehydratase
  • Carbonic Anhydrase (hpCA)
  • Carbonic Anhydrase (mtCA 1)
  • Carbonic Anhydrase (mtCA 3)
  • Carbonic Anhydrase 2 (Can2)
  • Carbonic Anhydrase III
  • Carbonic Anhydrase VA
  • Carbonic Anhydrase VB
  • Carbonic Anhydrase XV
  • Carbonic anhydrase
  • Carbonic anhydrase 1
  • Carbonic anhydrase 12
  • Carbonic anhydrase 2
  • Carbonic anhydrase 6 (CA-VI)
  • Carbonic anhydrase 7
  • Carbonic anhydrase 9
  • Carbonic anhydrase, alpha family
  • Delta carbonic anhydrase
  • beta-Carbonic Anhydrase
  • 4-methylbenzene-1-sulfonamide
  • CHEMBL574
  • aromatic/heteroaromatic sulfonamide 4
  • hCA inhibitor, 7
89 Ki 3 IC50 8 Kd
  • 5-hydroxytryptamine receptor 1A
  • 5-hydroxytryptamine receptor 2A
  • ADRA1A
  • ADRA1B
  • Adrenergic alpha1B
  • Adrenergic receptor
  • Adrenergic receptor alpha
  • Adrenergic receptor alpha-2
  • Alpha adrenergic receptor (1a and 1d)
  • Alpha adrenergic receptor 1A and 1B
  • Alpha adrenergic receptor 1A and 1D
  • Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor
  • Alpha-1A adrenergic receptor
  • Alpha-1D adrenergic receptor
  • Cerebral cortex alpha adrenergic receptor
  • D(2) dopamine receptor
  • D(3) dopamine receptor
  • Dopamine receptor
  • HTR2C
  • Serotonin (5-HT) receptor
  • Serotonin 1B/1D receptor
  • Serotonin 2 (5-HT2) receptor
  • 8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-azaspiro[4.5]decane-7,9-dione
  • 8-[2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl]-8-azaspiro[4.5]decane-7,9-dione
  • 8-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione
  • 8-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-8-aza-spiro[4.5]decane-7,9-dione(BMY-7378)
  • BMY 7378
  • BMY-7378
  • CHEMBL1256934
  • CHEMBL13647
  • CHEMBL543741
63 Ki 36 IC50 1 EC50
  • AGTR1
  • Acetylcholinesterase
  • Adenosine Kinase (AK)
  • Alpha-1A adrenergic receptor
  • Angiotensin II AT2
  • BDKRB2
  • Beta-2 adrenergic receptor
  • CCKBR
  • Calcium channel
  • Choline Acetyltransferase
  • Corticotropin-Releasing Factor
  • D(1A) dopamine receptor
  • EDNRA
  • EDNRB
  • Estrogen receptor
  • Fatty-acid amide hydrolase 1
  • GALANIN
  • GRIA3
  • Gamma-aminobutyric acid receptor subunit alpha-1
  • Gamma-aminobutyric acid type B receptor subunit 1
  • Glutamate receptor ionotropic, NMDA 1
  • Glutamate receptor ionotropic, kainate 1
  • Glutamic acid decarboxylase
  • Glycine
  • Glycine, non-strychnine
  • HRH3
  • Histamine H1 receptor
  • Histamine H2 receptor
  • Leukotriene B4
  • Leukotriene D4
  • Melatonin
  • Monoamine Oxidase Type B (MAO-B)
  • Monoamine oxidase
  • Mu-type opioid receptor
  • Muscarinic acetylcholine receptor M1
  • Muscarinic acetylcholine receptor M2
  • Neurokinin 1 receptor
  • Neurokinin 2 receptor
  • Neurokinin 3 receptor
  • Nitric-oxide synthase, brain
  • Norepinephrine transporter
  • Oxytocin receptor
  • PTAFR
  • Potassium Channel, Ca2+ Act., VI
  • Potassium voltage-gated channel subfamily H member 2
  • Renal Outer Medullary Potassium (ROMK)
  • Serotonin
  • Sigma non-opioid intracellular receptor 1
  • Small conductance calcium-activated potassium channel
  • Sodium (Site 1)
  • Sodium (Site 2)
  • Sodium-dependent dopamine transporter
  • TRH
  • Testosterone
  • Thromboxane A2 receptor
  • Transient receptor potential M8 protein (TRPM8)
  • Transient receptor potential cation channel subfamily A member 1
  • Transient receptor potential cation channel subfamily M member 8
  • Transient receptor potential cation channel subfamily M member 8 (TRPM8)
  • Transient receptor potential cation channel subfamily V member 1
  • VASOPRESSIN V1
  • VIP
  • Vanilloid receptor
  • Voltage-dependent N-type calcium channel subunit alpha-1B
  • adrenergic Alpha2
  • n-AChR
  • 4-(3-Chloro-pyridin-2-yl)-piperazine-1-carboxylic acid (4-tert-butyl-phenyl)-amide
  • BCTC
  • CHEMBL441472
  • N-(4-tert-butylphenyl)-4-(3-chloropyridin-2-yl)piperazine-1-carboxamide
100 IC50
  • 5'-AMP-activated protein kinase Complex 1
  • AMPK alpha2/beta1/gamma1
  • Activin receptor type-1B
  • Angiopoietin-1 receptor
  • Aurora kinase B
  • Axin-1/Glycogen synthase kinase-3 beta
  • Beta-adrenergic receptor kinase 1
  • CDK7/Cyclin H/MNAT1
  • CaM kinase IV
  • Casein kinase I isoform alpha
  • Casein kinase II subunit alpha
  • Cyclin-Dependent Kinase 5 (CDK5)
  • Cyclin-Dependent Kinase 9 (CDK9)
  • Cyclin-dependent kinase 2
  • Cytoplasmic tyrosine-protein kinase BMX
  • Death-associated protein kinase 1
  • Dual specificity mitogen-activated protein kinase kinase 1
  • Dual specificity mitogen-activated protein kinase kinase 6
  • Dual specificity protein kinase CLK2
  • Dual-specificity tyrosine-phosphorylation regulated kinase 1A
  • Ephrin receptor
  • Ephrin type-A receptor 3 (EPHA3)
  • Ephrin type-B receptor 2
  • Epidermal growth factor receptor
  • Fibroblast growth factor receptor 2
  • G protein-coupled receptor kinase 4
  • G protein-coupled receptor kinase 6
  • Glycogen synthase kinase-3
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Inhibitor of nuclear factor kappa-B kinase subunit beta
  • Inhibitor of nuclear factor kappa-B kinase subunit epsilon
  • Insulin receptor
  • Insulin-like growth factor I receptor
  • Interleukin-1 receptor-associated kinase 1
  • Interleukin-1 receptor-associated kinase 4
  • Leucine-rich repeat serine/threonine-protein kinase 2 (LRRK2)
  • Lysyl-tRNA synthetase
  • MAP kinase-activated protein kinase 2
  • MAP kinase-activated protein kinase 5
  • MAP/microtubule affinity-regulating kinase 4
  • Macrophage colony-stimulating factor 1 receptor (CSF1R)
  • Mast/stem cell growth factor receptor Kit
  • Mitogen-activated protein kinase 1
  • Mitogen-activated protein kinase 13 (MAPK13)
  • Mitogen-activated protein kinase 14
  • Mitogen-activated protein kinase 8
  • Mitogen-activated protein kinase 9
  • Mitogen-activated protein kinase kinase kinase 8
  • NT-3 growth factor receptor
  • NUAK family SNF1-like kinase 1
  • Non-receptor tyrosine-protein kinase TYK2
  • PAK 1/CDC42
  • PAS domain-containing serine/threonine-protein kinase
  • Phosphoinositide 3-Kinase (PI3K), delta
  • Protein kinase C (PKC)
  • Protein kinase C iota (PKCι)
  • Protein kinase C theta type
  • Protein kinase N1
  • Proto-oncogene tyrosine-protein kinase Src
  • RAC-alpha serine/threonine-protein kinase
  • Receptor tyrosine-protein kinase erbB-2
  • Rho-associated protein kinase 1
  • Rho-associated protein kinase 2
  • Ribosomal protein S6 kinase (P70S6K)
  • Ribosomal protein S6 kinase alpha-3
  • Serine/threonine-protein kinase AKT
  • Serine/threonine-protein kinase AKT2
  • Serine/threonine-protein kinase B-raf
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase Chk2
  • Serine/threonine-protein kinase MRCK-A
  • Serine/threonine-protein kinase MST4
  • Serine/threonine-protein kinase NEK6
  • Serine/threonine-protein kinase Nek2
  • Serine/threonine-protein kinase Nek4
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase SRPK1
  • Serine/threonine-protein kinase Sgk1
  • Serine/threonine-protein kinase TAO2
  • Serine/threonine-protein kinase TBK1
  • Serine/threonine-protein kinase c-TAK1
  • Serine/threonine-protein kinase pim-1
  • Sphingosine kinase 1 (SPHK1)
  • Testis-specific serine/threonine-protein kinase 1
  • Tyrosine-protein kinase ABL1
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase BTK
  • Tyrosine-protein kinase HCK
  • Tyrosine-protein kinase ITK/TSK
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase Lck
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor FLT3
  • Vascular endothelial growth factor receptor 2
  • Voltage-gated potassium channel subunit Kv7.1/Misshapen-like kinase 1
  • [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
  • cAMP-dependent protein kinase (PKA)
  • CHEMBL3884319
100 IC50
  • 3-phosphoinositide dependent protein kinase-1
  • 5'-AMP-activated protein kinase Complex 1
  • Activin receptor type-1B
  • Aurora kinase A/B
  • Axin-1/Glycogen synthase kinase-3 beta
  • BRAF/CRAF
  • CaM kinase IV
  • Calmodulin/Proto-oncogene tyrosine-protein kinase Src
  • Casein kinase I isoform alpha
  • Casein kinase II subunit alpha
  • Cereblon/BCR/ABL
  • Cyclin-Dependent Kinase 5 (CDK5)
  • Cyclin-Dependent Kinase 9 (CDK9)
  • Cyclin-dependent kinase 2
  • Cyclin-dependent kinase 7
  • Cytoplasmic tyrosine-protein kinase BMX
  • Death-associated protein kinase 1
  • Dual specificity mitogen-activated protein kinase kinase 1/Mitogen-activated protein kinase 1/RAF proto-oncogene serine/threonine-protein kinase
  • Dual specificity mitogen-activated protein kinase kinase 6
  • Dual specificity protein kinase CLK2
  • Dual-specificity tyrosine-phosphorylation regulated kinase 1A
  • Ephrin receptor
  • Ephrin type-A receptor 3 (EPHA3)
  • Ephrin type-B receptor 2
  • Epidermal growth factor receptor
  • Fibroblast growth factor receptor 2
  • G protein-coupled receptor kinase 4
  • G protein-coupled receptor kinase 6
  • G-protein coupled receptor kinase 2
  • Glycogen synthase kinase-3
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Inhibitor of NF-kappa-B kinase alpha/beta
  • Inhibitor of nuclear factor kappa-B kinase subunit epsilon
  • Insulin receptor
  • Insulin-like growth factor I receptor
  • Interleukin-1 receptor-associated kinase 1
  • Interleukin-1 receptor-associated kinase 4
  • Leucine-rich repeat serine/threonine-protein kinase 2
  • MAP kinase-activated protein kinase 2
  • MAP kinase-activated protein kinase 5
  • MAP/microtubule affinity-regulating kinase 3
  • MAP/microtubule affinity-regulating kinase 4
  • Macrophage colony-stimulating factor 1 receptor (CSF1R)
  • Mast/stem cell growth factor receptor Kit
  • Mitogen-activated protein kinase 14
  • Mitogen-activated protein kinase 8
  • Mitogen-activated protein kinase 9
  • NT-3 growth factor receptor
  • NUAK family SNF1-like kinase 1
  • Non-receptor tyrosine-protein kinase TYK2
  • PAK 1/CDC42
  • PAS domain-containing serine/threonine-protein kinase
  • Phosphoinositide 3-Kinase (PI3K), delta
  • Protein kinase C iota type/zeta type
  • Protein kinase C theta type
  • Protein kinase N1
  • RAC-alpha serine/threonine-protein kinase
  • RAF proto-oncogene serine/threonine-protein kinase
  • Receptor tyrosine-protein kinase erbB-2
  • Rho-associated protein kinase 1
  • Rho-associated protein kinase 2
  • Ribosomal protein S6 kinase (P70S6K)
  • Ribosomal protein S6 kinase alpha-1/alpha-3
  • Serine/threonine-protein kinase AKT
  • Serine/threonine-protein kinase AKT2
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase MRCK-A
  • Serine/threonine-protein kinase MST4
  • Serine/threonine-protein kinase NEK2
  • Serine/threonine-protein kinase NEK6
  • Serine/threonine-protein kinase Nek4
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase SRPK1
  • Serine/threonine-protein kinase Sgk1
  • Serine/threonine-protein kinase TAO2
  • Serine/threonine-protein kinase TBK1
  • Serine/threonine-protein kinase pim-1
  • Sphingosine kinase 1
  • Testis-specific serine/threonine-protein kinase 1
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase BTK
  • Tyrosine-protein kinase HCK
  • Tyrosine-protein kinase ITK/TSK
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase Lck
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor FLT3
  • Vascular endothelial growth factor receptor 2
  • Vascular endothelial growth factor receptor 2 and tyrosine-protein kinase TIE-2 (KDR and TIE2)
  • Voltage-gated potassium channel subunit Kv7.1/Misshapen-like kinase 1
  • cAMP-dependent protein kinase (PKA)
  • p38 delta/gamma
  • CHEMBL4569508
100 IC50
  • 3-phosphoinositide dependent protein kinase-1
  • 5'-AMP-activated protein kinase Complex 1
  • Activin receptor type-1B
  • Aurora kinase A/B
  • Axin-1/Glycogen synthase kinase-3 beta
  • BRAF/CRAF
  • CaM kinase IV
  • Calmodulin/Proto-oncogene tyrosine-protein kinase Src
  • Casein kinase I isoform alpha
  • Casein kinase II subunit alpha
  • Cereblon/BCR/ABL
  • Cyclin-Dependent Kinase 5 (CDK5)
  • Cyclin-Dependent Kinase 9 (CDK9)
  • Cyclin-dependent kinase 2
  • Cyclin-dependent kinase 7
  • Cytoplasmic tyrosine-protein kinase BMX
  • Death-associated protein kinase 1
  • Dual specificity mitogen-activated protein kinase kinase 1/Mitogen-activated protein kinase 1/RAF proto-oncogene serine/threonine-protein kinase
  • Dual specificity mitogen-activated protein kinase kinase 6
  • Dual specificity protein kinase CLK2
  • Dual-specificity tyrosine-phosphorylation regulated kinase 1A
  • Ephrin receptor
  • Ephrin type-A receptor 3 (EPHA3)
  • Ephrin type-B receptor 2
  • Epidermal growth factor receptor
  • Fibroblast growth factor receptor 2
  • G protein-coupled receptor kinase 4
  • G protein-coupled receptor kinase 6
  • G-protein coupled receptor kinase 2
  • Glycogen synthase kinase-3
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Inhibitor of NF-kappa-B kinase alpha/beta
  • Inhibitor of nuclear factor kappa-B kinase subunit epsilon
  • Insulin receptor
  • Insulin-like growth factor I receptor
  • Interleukin-1 receptor-associated kinase 1
  • Interleukin-1 receptor-associated kinase 4
  • Leucine-rich repeat serine/threonine-protein kinase 2
  • MAP kinase-activated protein kinase 2
  • MAP kinase-activated protein kinase 5
  • MAP/microtubule affinity-regulating kinase 3
  • MAP/microtubule affinity-regulating kinase 4
  • Macrophage colony-stimulating factor 1 receptor (CSF1R)
  • Mast/stem cell growth factor receptor Kit
  • Mitogen-activated protein kinase 14
  • Mitogen-activated protein kinase 8
  • Mitogen-activated protein kinase 9
  • NT-3 growth factor receptor
  • NUAK family SNF1-like kinase 1
  • Non-receptor tyrosine-protein kinase TYK2
  • PAK 1/CDC42
  • PAS domain-containing serine/threonine-protein kinase
  • Phosphoinositide 3-Kinase (PI3K), delta
  • Protein kinase C iota type/zeta type
  • Protein kinase C theta type
  • Protein kinase N1
  • RAC-alpha serine/threonine-protein kinase
  • RAF proto-oncogene serine/threonine-protein kinase
  • Receptor tyrosine-protein kinase erbB-2
  • Rho-associated protein kinase 1
  • Rho-associated protein kinase 2
  • Ribosomal protein S6 kinase (P70S6K)
  • Ribosomal protein S6 kinase alpha-1/alpha-3
  • Serine/threonine-protein kinase AKT
  • Serine/threonine-protein kinase AKT2
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase MRCK-A
  • Serine/threonine-protein kinase MST4
  • Serine/threonine-protein kinase NEK2
  • Serine/threonine-protein kinase NEK6
  • Serine/threonine-protein kinase Nek4
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase SRPK1
  • Serine/threonine-protein kinase Sgk1
  • Serine/threonine-protein kinase TAO2
  • Serine/threonine-protein kinase TBK1
  • Serine/threonine-protein kinase pim-1
  • Sphingosine kinase 1
  • Testis-specific serine/threonine-protein kinase 1
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase BTK
  • Tyrosine-protein kinase HCK
  • Tyrosine-protein kinase ITK/TSK
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase Lck
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor FLT3
  • Vascular endothelial growth factor receptor 2
  • Vascular endothelial growth factor receptor 2 and tyrosine-protein kinase TIE-2 (KDR and TIE2)
  • Voltage-gated potassium channel subunit Kv7.1/Misshapen-like kinase 1
  • cAMP-dependent protein kinase (PKA)
  • p38 delta/gamma
  • CHEMBL4550702
100 IC50
  • 3-phosphoinositide dependent protein kinase-1
  • 5'-AMP-activated protein kinase Complex 1
  • Activin receptor type-1B
  • Aurora kinase A/B
  • Axin-1/Glycogen synthase kinase-3 beta
  • BRAF/CRAF
  • CaM kinase IV
  • Calmodulin/Proto-oncogene tyrosine-protein kinase Src
  • Casein kinase I isoform alpha
  • Casein kinase II subunit alpha
  • Cereblon/BCR/ABL
  • Cyclin-Dependent Kinase 5 (CDK5)
  • Cyclin-Dependent Kinase 9 (CDK9)
  • Cyclin-dependent kinase 2
  • Cyclin-dependent kinase 7
  • Cytoplasmic tyrosine-protein kinase BMX
  • Death-associated protein kinase 1
  • Dual specificity mitogen-activated protein kinase kinase 1/Mitogen-activated protein kinase 1/RAF proto-oncogene serine/threonine-protein kinase
  • Dual specificity mitogen-activated protein kinase kinase 6
  • Dual specificity protein kinase CLK2
  • Dual-specificity tyrosine-phosphorylation regulated kinase 1A
  • Ephrin receptor
  • Ephrin type-A receptor 3 (EPHA3)
  • Ephrin type-B receptor 2
  • Epidermal growth factor receptor
  • Fibroblast growth factor receptor 2
  • G protein-coupled receptor kinase 4
  • G protein-coupled receptor kinase 6
  • G-protein coupled receptor kinase 2
  • Glycogen synthase kinase-3
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Inhibitor of NF-kappa-B kinase alpha/beta
  • Inhibitor of nuclear factor kappa-B kinase subunit epsilon
  • Insulin receptor
  • Insulin-like growth factor I receptor
  • Interleukin-1 receptor-associated kinase 1
  • Interleukin-1 receptor-associated kinase 4
  • Leucine-rich repeat serine/threonine-protein kinase 2
  • MAP kinase-activated protein kinase 2
  • MAP kinase-activated protein kinase 5
  • MAP/microtubule affinity-regulating kinase 3
  • MAP/microtubule affinity-regulating kinase 4
  • Macrophage colony-stimulating factor 1 receptor (CSF1R)
  • Mast/stem cell growth factor receptor Kit
  • Mitogen-activated protein kinase 14
  • Mitogen-activated protein kinase 8
  • Mitogen-activated protein kinase 9
  • NT-3 growth factor receptor
  • NUAK family SNF1-like kinase 1
  • Non-receptor tyrosine-protein kinase TYK2
  • PAK 1/CDC42
  • PAS domain-containing serine/threonine-protein kinase
  • Phosphoinositide 3-Kinase (PI3K), delta
  • Protein kinase C iota type/zeta type
  • Protein kinase C theta type
  • Protein kinase N1
  • RAC-alpha serine/threonine-protein kinase
  • RAF proto-oncogene serine/threonine-protein kinase
  • Receptor tyrosine-protein kinase erbB-2
  • Rho-associated protein kinase 1
  • Rho-associated protein kinase 2
  • Ribosomal protein S6 kinase (P70S6K)
  • Ribosomal protein S6 kinase alpha-1/alpha-3
  • Serine/threonine-protein kinase AKT
  • Serine/threonine-protein kinase AKT2
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase MRCK-A
  • Serine/threonine-protein kinase MST4
  • Serine/threonine-protein kinase NEK2
  • Serine/threonine-protein kinase NEK6
  • Serine/threonine-protein kinase Nek4
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase SRPK1
  • Serine/threonine-protein kinase Sgk1
  • Serine/threonine-protein kinase TAO2
  • Serine/threonine-protein kinase TBK1
  • Serine/threonine-protein kinase pim-1
  • Sphingosine kinase 1
  • Testis-specific serine/threonine-protein kinase 1
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase BTK
  • Tyrosine-protein kinase HCK
  • Tyrosine-protein kinase ITK/TSK
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase Lck
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor FLT3
  • Vascular endothelial growth factor receptor 2
  • Vascular endothelial growth factor receptor 2 and tyrosine-protein kinase TIE-2 (KDR and TIE2)
  • Voltage-gated potassium channel subunit Kv7.1/Misshapen-like kinase 1
  • cAMP-dependent protein kinase (PKA)
  • p38 delta/gamma
  • CHEMBL4552628