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Compound Name:

Compounds Sorted by Binding Data per Compound

1   2   3   4   5   6   7   8   9   10   11   12   13   14   15   16   17   18   19   20   21   
22   23   24   25   26   27   28   29   30   31   32   33   34   35   36   37   38   39   40   41   42   
43   44   45   46   47   48   49   50   51   52   53   54   55   56   57   58   59   60   61   62   63   
64   65   66   67   68   69   70   71   72   73   74   75   76   77   78   79   80   81   82   83   84   
85   86   87   88   89   90   91   92   93   94   95   96   97   98   99   100   101   102   103   104   105   
106   107   108   109   110   111   112   113   114   115   116   117   118   119   120   121   122   123   124   125   127   
128   129   130   132   133   134   135   136   137   138   139   140   141   143   144   145   146   147   148   149   150   
151   153   154   155   156   159   160   161   163   164   165   168   170   171   173   174   176   178   179   183   184   
186   188   189   190   191   192   193   196   198   199   200   203   205   206   207   208   209   210   216   220   224   
226   227   230   232   237   238   241   243   248   252   253   259   261   270   274   276   277   285   291   303   304   
313   318   323   325   328   333   335   337   339   341   353   360   361   365   389   393   398   401   413   433   442   
444   445   446   447   448   451   453   454   455   457   458   460   463   465   467   473   477   478   482   484   499   
504   505   506   517   525   543   549   551   554   591   606   663   691   708   796   804   821   825   833   842   847   
854   855   861   873   879   883   887   913   914   925   926   938   947   1010   1027   1050   1052   1081   1082   1102   1115   
1130   1133   1206   1262   1543   1639   1903   2029   

Compounds Sorted Alphabetically

Compound Name (alphabetical)	Enz. Inhib. Data							ITC Data	Binding Targets	Alternate Compound Names
	Ki	IC50	Kd	EC50	Koff	Kon	Other
BDBM18224	5	108	0	0	0	0	0	0	Bacterial dihydrofolate reductase DHFR Dihydrofolate Reductase (DHFR) Dihydrofolate reductase Dihydrofolate reductase (DHFR) Protein Wnt-3a Zinc finger protein GLI1	6-[(2,5-dimethoxyphenyl)methyl]-5-methylpyrido[2,3-d]pyrimidine-2,4-diamine CHEMBL7492 PTX Piritrexim [2-amino-6-(2,5-dimethoxybenzyl)-5-methyl-pyrido[2,3-d]pyrimidin-4-yl]amine;2-hydroxyethanesulfonic acid
BDBM50463483	112	1	0	0	0	0	0	0	Aurora kinase A/Targeting protein for Xklp2 Aurora kinase B Axin-1/Glycogen synthase kinase-3 beta BR serine/threonine-protein kinase 1 BR serine/threonine-protein kinase 2 CAMK2A CAMK2B CaM kinase I delta CaM kinase IV Casein kinase I isoform alpha Ceramide kinase Choline kinase alpha Citron Rho-interacting kinase Cyclin-Dependent Kinase 1 (CDK1) Cyclin-Dependent Kinase 2 (CDK2) Cyclin-Dependent Kinase 5 (CDK5) Cytochrome P450 3A Cytoplasmic tyrosine-protein kinase BMX DNA-dependent protein kinase Death-associated protein kinase 1 Dual specificity protein kinase CLK3 Dual-specificity tyrosine-phosphorylation regulated kinase 1A Dual-specificity tyrosine-phosphorylation regulated kinase 2 Ephrin receptor Ephrin type-B receptor 2 Ephrin type-B receptor 4 Epidermal growth factor receptor Fibroblast growth factor receptor 1 Fibroblast growth factor receptor 2 Fibroblast growth factor receptor 3 Fibroblast growth factor receptor 4 Focal adhesion kinase 1 Focal adhesion kinase 1/vascular endothelial growth factor receptor 3 Hepatocyte growth factor receptor Insulin receptor Insulin-like growth factor I receptor Interleukin-1 receptor-associated kinase 1 Interleukin-1 receptor-associated kinase 4 MAP kinase-activated protein kinase 2 Macrophage colony stimulating factor receptor Macrophage-stimulating protein receptor Mast/stem cell growth factor receptor Kit Mitogen-activated protein kinase 1 Mitogen-activated protein kinase 10 Mitogen-activated protein kinase 12 Mitogen-activated protein kinase kinase kinase 14 Mitogen-activated protein kinase kinase kinase 8 Mitogen-activated protein kinase kinase kinase kinase 4 PAK 1/CDC42 PAS domain-containing serine/threonine-protein kinase PKC alpha and beta-2 PTK2B protein tyrosine kinase 2 beta (PTK2B) Phosphorylase kinase Platelet-derived growth factor receptor Protein kinase C, PKC; classical/novel Proto-oncogene tyrosine-protein kinase ROS Proto-oncogene tyrosine-protein kinase Src Proto-oncogene tyrosine-protein kinase receptor Ret RAC-alpha serine/threonine-protein kinase Rho-associated protein kinase 1 Ribosomal protein S6 kinase Ribosomal protein S6 kinase alpha 1 Ribosomal protein S6 kinase alpha 2 Ribosomal protein S6 kinase alpha 4 Ribosomal protein S6 kinase alpha-1/alpha-3 Serine/threonine-protein kinase 4 (STK4) Serine/threonine-protein kinase AKT Serine/threonine-protein kinase AKT2 Serine/threonine-protein kinase ATR Serine/threonine-protein kinase Aurora-C Serine/threonine-protein kinase Chk1/2 Serine/threonine-protein kinase D2 Serine/threonine-protein kinase DCLK1 Serine/threonine-protein kinase DCLK2 Serine/threonine-protein kinase MARK1 Serine/threonine-protein kinase NEK2 Serine/threonine-protein kinase Nek1 Serine/threonine-protein kinase PAK 2 Serine/threonine-protein kinase Sgk1 Serine/threonine-protein kinase Sgk2 Serine/threonine-protein kinase Sgk3 Serine/threonine-protein kinase TBK1 Serine/threonine-protein kinase c-TAK1 Serine/threonine-protein kinase pim-1 Serine/threonine-protein kinase pim-2 Sphingosine kinase 1 Testis-specific serine/threonine-protein kinase 2 Tyrosine-protein kinase ABL1 Tyrosine-protein kinase BTK Tyrosine-protein kinase CSK Tyrosine-protein kinase FER Tyrosine-protein kinase Fyn Tyrosine-protein kinase HCK Tyrosine-protein kinase JAK3 Tyrosine-protein kinase Lck Tyrosine-protein kinase Lyn Tyrosine-protein kinase Mer Tyrosine-protein kinase SYK Tyrosine-protein kinase Yes Tyrosine-protein kinase ZAP-70 Tyrosine-protein kinase receptor FLT3 Tyrosine-protein kinase receptor TYRO3 Vascular endothelial growth factor receptor 1 Vascular endothelial growth factor receptor 2 Vascular endothelial growth factor receptor 2 and tyrosine-protein kinase TIE-2 (KDR and TIE2) Voltage-gated potassium channel subunit Kv7.1/Misshapen-like kinase 1 p21-Activated kinase 3 (PAK3) p38 delta/gamma	CHEMBL4245242